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N-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[(3R)-piperidin-3-yl]piperidin-4-amine
(3R,4R)-4-ethyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine-3,4-diol
2-(2,5-dioxoimidazolidin-1-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
N-{[(2S,4S)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-fluoropyrrolidin-2-yl]methyl}acetamide
4-chloro-3-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)-N-methylbenzamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(cyclohex-1-en-1-yl)ethan-1-one
N-(1-methyl-1H-pyrazol-4-yl)-5-[1-(3-methylfuran-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-amino-6-(2,2-dimethylcyclopropyl)-4-[2-(ethylamino)pyrimidin-5-yl]-5-methylpyridine-3-carbonitrile
1-phenyl-4-(2-propoxypropanoyl)piperazin-2-one
4-[6-(2-fluoro-4-methylphenyl)pyridine-3-carbonyl]morpholine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
[(3-chloro-2,6-difluorophenyl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N,1-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
5-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-[(2E)-4-methylpent-2-en-1-yl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
N-(4-methyl-1-propyl-1H-pyrazol-5-yl)-2-(4-{thieno[2,3-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)acetamide
5-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
6-methyl-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-acetamido-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
(2S,4S)-N-ethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-[(3-methoxyphenyl)methyl]-3-(3-methylthiophen-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-1-[4-(oxolan-2-ylmethoxy)phenyl]-3-(thiophen-3-ylmethyl)urea
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}cyclobutanamine
N-methyl-2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-amine
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
4-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]methyl}morpholine
(2,1,3-benzothiadiazol-5-ylmethyl)({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-phenylpiperazin-2-one
5-methoxy-1-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-indole-2-carboxamide
[5-chloro-7-(2-methyl-5-propylpyrimidin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-(4-hydroxyphenyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
N-(5-methyl-2,1,3-benzothiadiazol-4-yl)-2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carboxamide
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(3-fluorobenzoyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
N-[2-(dimethylamino)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
7-cyclopentyl-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoacetamide
N-[(3,5-difluorophenyl)methyl]-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(6-methoxypyrimidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
N3-methyl-N5-[(3-methylphenyl)methyl]-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-[2-(dimethylamino)ethyl]-8-(quinolin-4-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(1-methylpyrrolidin-3-yl)-9-(3-phenylpropyl)-2,9-diazaspiro[5.5]undecan-3-one
2,8-dimethyl-3-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}quinoline
5-[3-(2-methylphenoxy)azetidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(3-phenoxyphenyl)methyl]amine