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1-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[3-(2-methoxyphenyl)propyl]-1,2,3,4-tetrahydronaphthalen-2-amine
2-(oxolan-2-ylmethoxy)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N4-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-(2-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-2-yl}ethyl)morpholine
2-(2-chlorophenoxy)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(3-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
3-{2-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
4-[3-(2-benzylmorpholine-4-carbonyl)phenyl]morpholine
1-[1-(3-hydroxypyridine-2-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
{5-[3-(3-fluorophenoxymethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methanol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
5-[({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
ethyl 5-{3-tert-butyl-1-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
4-{[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]amino}pyrimidine-5-carboxylic acid
1-{[4-(difluoromethoxy)phenyl]methyl}-3-(3,4-dimethoxybenzoyl)piperidine
3-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)pyridine
N3-[(1-hydroxycyclohexyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-hydroxy-N-[3-hydroxy-1-(4-methylphenyl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
8-(4-methylpentyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(2R,3S,6R)-5-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-(2,3,4-trifluorophenyl)ethan-1-one
1-cyclopentyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
(4aR,7aS)-1-(2-methoxyacetyl)-4-(quinoxaline-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopropyl-5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]pyrimidine
(5S,9aS,9bS)-5-(3-phenoxyphenyl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(4-{2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazol-2-yl)pyridine
2-methyl-6-{1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-4-yl}pyrimidin-4-ol
N-cyclopropyl-1-{2-[1-(3,4-dimethoxybenzenesulfonyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-cyclopentyl-3-cyclopropyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrazole-5-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]thiophene-3-sulfonamide
N-benzyl-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-[(4-methoxyphenyl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
methyl 5-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-5-oxopentanoate
{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-methyl-N,2-bis(propan-2-yl)-1,3-thiazole-5-carboxamide
1-{2-oxo-2-[2-(3-phenylpropyl)morpholin-4-yl]ethyl}pyrrolidin-2-one
N-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(2-fluorophenyl)methyl]piperidin-3-amine
1-{2-methyl-3-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]propyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
2-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{1-[(dimethyl-1,3-thiazol-2-yl)methyl]-1H-imidazol-2-yl}-2-[(dimethylamino)methyl]phenol
N-[1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazole-4-carboxamide
[(3-methoxyphenyl)methyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2,6-dihydroxy-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
5-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)pyrimidin-2-amine
2-amino-3-ethyl-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[(2,4-difluorophenyl)methyl]-3-(3,4-dimethoxybenzoyl)piperidine
5-(2-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione