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2-ethyl-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridin-4-one
2-methyl-6-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]pyrimidin-4-ol
6-methyl-1-{3-oxo-3-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}-1,2-dihydropyridin-2-one
6-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
6-{[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]methyl}-1,4-oxazepan-6-ol
N-[(2-methoxyphenyl)methyl]-5-methyl-N-(pyridin-3-ylmethyl)pyridine-3-carboxamide
[(4-fluoro-3-methoxyphenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
4-[5-(2-propyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridine
2-{3-cyclopentyl-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazol-1-yl}acetic acid
(2S,4R)-4-amino-1-(2-cyclopentylacetyl)-N,N-diethylpyrrolidine-2-carboxamide
N-[1-({methyl[1-(thiophen-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-[(1R)-1-cyclohexylethyl]urea
1-tert-butyl-4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
2,2,2-trifluoro-N-(2-{[3-(propan-2-yl)-1,2-oxazol-5-yl]formamido}ethyl)acetamide
4-methyl-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-propyl-1H-pyrazole-5-carboxamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-5-(methoxymethyl)furan-2-carboxamide
4-{5-methyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
3-(cyclohexylamino)-N-[3-(1H-imidazol-1-yl)propyl]-5-(pyrrolidine-1-sulfonyl)benzamide
N-cyclopropyl-6-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-(2-benzyl-1,3-thiazole-4-carbonyl)-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
4-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]pyrazin-2-ol
1-(2-chlorophenyl)-4-[2-(4-fluorophenyl)-2-hydroxyacetyl]piperazin-2-one
(3S)-1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-amine
7-({2-[3-(dimethylamino)-2-hydroxypropoxy]-5-methoxyphenyl}methyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
methyl({[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
2-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
(3R,4R)-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-oxazole-4-carboxamide
1-(2-{[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}ethyl)piperidin-3-ol
9-[2-(propan-2-ylsulfanyl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
5-(2-fluoro-5-methylphenyl)-1-methyl-1H-[1,2,3]triazolo[4,5-b]pyridine
1-(2,2-dimethylpropyl)-3-hydroxy-3-[(4-propyl-1,4-diazepan-1-yl)methyl]piperidin-2-one
1-(2,5-dimethoxyphenyl)-3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}urea
{[3-(2-methylphenyl)phenyl]methyl}({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
2-ethoxy-5-(pyrimidin-5-yl)benzamide
5-(methoxymethyl)-3-methyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazole
1-{2-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]phenyl}ethan-1-one
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-2-sulfonyl)piperidine
N-(1,4-dioxan-2-ylmethyl)-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-({7-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
1-({1-[6-(4-hydroxyphenyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-(2-chloro-4-fluorobenzenesulfonyl)-4-[(dimethylamino)methyl]azepan-4-ol
5-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-4-methyl-2-(pyridin-3-yl)pyrimidine
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]propanamide