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1-(4-benzylpiperidin-1-yl)-3-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]propan-1-one
[(4-{2-[4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
3-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
4-(1H-imidazol-1-yl)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidine-4-carboxylic acid
N-(3,4-difluorophenyl)-5-{4-hydroxy-1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
(3R,4R)-1-{[3-(methylsulfanyl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
3-{5-[2-(diethylamino)ethyl]-1,3,4-thiadiazol-2-yl}-1-(oxan-2-ylmethyl)urea
(2R,3R,6R)-5-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]urea
1-{1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}piperidin-4-ol
2-(furan-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4R)-1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-ethyl-N-phenylpiperidin-3-amine
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(3-methylphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
6-({[1-(hydroxymethyl)cyclopentyl]methyl}amino)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
(2S,4R)-1-(1H-imidazol-4-ylmethyl)-N-(propan-2-yl)-4-[2-(pyridin-3-yl)acetamido]pyrrolidine-2-carboxamide
5-{1-butyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-2-methylpyrimidine
3-methoxy-1-{2-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
5-[(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
[3-(cyclopropylmethyl)-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-3-yl]methanol
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
7-(2-methyl-4-phenylpyridine-3-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
5-methyl-1-[(3-methylpyridin-4-yl)methyl]-5-phenylpiperidin-2-one
N-[(3S,4R)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
ethyl 4-[4-(hydroxymethyl)-4-(oxan-2-ylmethyl)piperidin-1-yl]piperidine-1-carboxylate
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
[3-(4-fluorophenoxy)propyl](methyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
4-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpent-4-enamide
1-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-3-methylpentan-1-one
5-cyclobutanecarbonyl-1'-(pyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-[(2S)-2-hydroxypropanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(morpholin-4-yl)ethyl]-4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)benzamide
2-[methyl(5-{[4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazin-1-yl]methyl}pyrimidin-2-yl)amino]acetic acid
4-(1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)phenol
N-[4-(1-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-imidazol-2-yl)phenyl]acetamide
2-[(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
(dicyclopropylmethyl)({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-({1-[2-(2-methoxyphenyl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
methyl 5-[(4-methylphenyl)methanesulfonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
(2S,4S)-4-amino-N,N-diethyl-1-[2-(6-methyl-1-benzofuran-3-yl)acetyl]pyrrolidine-2-carboxamide
5-methyl-1-{2-oxo-2-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(thiophen-2-ylmethyl)piperidine-3,5-dicarboxamide
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-4-(4H-1,2,4-triazol-4-yl)benzamide
2-[(4-methoxyphenyl)methyl]-4-(pyrrolidine-1-sulfonyl)morpholine
5-(3-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide