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N-(2,3-dihydro-1H-inden-2-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
2-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-2-yl}pyridine
(2S,4R)-4-(furan-2-amido)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
1,2-dimethyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indol-5-ol
N,3,5-trimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-indole-2-carboxamide
propan-2-yl 2-chloro-5-(4H-1,2,4-triazol-4-yl)benzoate
methyl 3-{1-[1-(methylcarbamoyl)propyl]-4-phenyl-1H-imidazol-5-yl}benzoate
1-[(diethylcarbamoyl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
7-chloro-N,3,5-trimethyl-N-[1-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
4-methyl-N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]pyrimidin-2-amine
3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-N-methylpyridin-2-amine
3-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-(4-hydroxyphenyl)-N-[(1S,2R)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]amino}cyclobutyl]acetamide
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(thian-4-yl)piperazine
4-(2-methoxyphenoxy)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
4-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-2-methyl-6-(1H-pyrazol-1-yl)pyrimidine
methyl 2-{4-[2-(benzyloxy)ethyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
N-methyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyridin-2-amine
3-(2-chlorophenyl)-1-{[1-(propan-2-yl)piperidin-3-yl]methyl}urea
N-(butan-2-yl)-N-(pyridin-4-ylmethyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-3-phenyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]acetamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-(1,2-oxazol-3-ylmethyl)urea
2-(morpholin-4-yl)-N-[2-(morpholin-4-yl)ethyl]-6-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}pyridine-3-carboxamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(4-methyl-1,3-oxazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-methyl-3-[2-(4-phenylpiperidin-1-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
ethyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
1-[2-(cyclopentylcarbamoyl)ethyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-(furan-2-yl)-5-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
(3aS,6aS)-2-cyclopropanecarbonyl-5-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-(1H-imidazol-1-yl)propyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
3-(5-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
1-{[2-(difluoromethoxy)phenyl]methyl}-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
6-methyl-4-oxo-N-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(cyclohexylmethyl)-N-[2-(diethylamino)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-methylfuran-2-carboxamide
(3S,9aR)-8-{[3-(methylsulfanyl)phenyl]methyl}-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
(1R,2R)-2-[5-methyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,3-dimethylpiperazin-2-one
ethyl 4-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
2-ethoxy-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
4-{2-[4-(dimethylamino)phenyl]acetyl}-1-(2-methylphenyl)piperazin-2-one
2-[1-cyclopropyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]acetamide
N-[(2,5-dimethylphenyl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-ethoxy-3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one