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4-methyl-6-(4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-1-yl)pyrimidin-2-amine
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-(1-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-2-one
N'-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-N-(5-methyl-1,2-oxazol-3-yl)ethanediamide
3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methyl-1-(2-methyl-5-sulfamoylphenyl)urea
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
3-(azepane-1-carbonyl)-N-(3-methylbutyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2,3-dihydro-1H-indene-1-carboxamide
2-ethyl-9-{2-methylthieno[3,2-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
3-[(4-fluorophenyl)formamido]-N-[1-(methoxymethyl)cyclopropyl]-N-methylpropanamide
N-[2-(2,5-dimethylphenoxy)ethyl]-6-(2-hydroxyethyl)-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(hydroxymethyl)-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-ol
N-({1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
4-(4-chlorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]butanamide
2-{5-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
3-(2-methyl-1H-imidazol-1-yl)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
5-({[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl](methyl)amino}methyl)-2-methoxyphenol
N-[2-(methylsulfanyl)phenyl]-4-(oxan-4-yl)piperazine-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-(1,3-benzothiazol-2-yl)-4-cyclopropanecarbonyl-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-4-ethyl-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-5-carboxamide
2-methyl-4-{3-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]phenyl}butan-2-ol
3-(2H-1,3-benzodioxol-5-yl)-5-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-cyclopropyl-2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}acetamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5,6-dimethylpyrimidin-4-amine
7-methoxy-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(2-methoxyethyl)-9-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(3-fluorophenyl)ethyl]-1-(1-methylcyclopropanecarbonyl)piperidine
3-[(3R,4S)-1-(2-methoxy-6-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
6-[(1-acetylpiperidin-4-yl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-(2,2,7-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
methyl (2S,4R)-1-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-4-hydroxypyrrolidine-2-carboxylate
6-(dimethylamino)-N-[2-(1H-imidazol-4-yl)ethyl]pyridine-3-carboxamide
3-{[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
methyl 4-[({[4-(dimethylamino)oxan-4-yl]methyl}carbamoyl)amino]benzoate
3-methyl-7-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 4-[2-amino-3-cyano-6-(5-methylfuran-2-yl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
N-ethyl-5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]pyrimidin-2-amine
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-benzylmorpholin-2-yl)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-[3-(furan-2-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
6-(dimethyl-1,2-oxazol-4-yl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
6-(4-aminoazepane-1-carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3,6-dimethyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1-benzofuran-2-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
5-[(adamantan-1-ylsulfanyl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[1'-(2-hydroxy-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
4-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-[(3-methoxyphenyl)methyl]morpholine
5-[1-(1,3-benzothiazole-5-carbonyl)pyrrolidin-2-yl]-N,N-dimethylthiophene-2-carboxamide