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5-{[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole
4-{1-[(methylcarbamoyl)methyl]piperidin-3-yl}benzoic acid
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(naphthalen-1-yl)ethyl]butanamide
4-{5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazine-1-carbaldehyde
1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propane-1,2-dione
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-(cyclopropylmethyl)-N-(propan-2-yl)acetamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]ethan-1-one
N-[(3-chlorophenyl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-methyl-1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidine-3-carboxamide
3-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propane-1,2-diol
1-(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[1-(thiophen-2-yl)ethyl]acetamide
methyl 3-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}-5-methoxybenzoate
4-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine-3-carbonyl)morpholine
4-[(2,4-difluorophenyl)methyl]-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
8-[2-(4-methanesulfonylphenyl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-5-hydroxypyrazine-2-carboxamide
{4-[(5-benzyl-4-phenyl-1H-imidazol-1-yl)methyl]oxan-4-yl}methanol
(3aR,6aS)-2-methyl-5-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
1-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
N-(3-methoxypropyl)-6,6-dimethyl-N-[(4-methylphenyl)methyl]-5-oxothiomorpholine-3-carboxamide
1-[4-(2-ethoxyethyl)-6-hydroxy-1,4-diazepan-1-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
ethyl 1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
3-(2,5,7-trimethylquinoline-4-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
3-[1-(1,3-benzothiazole-6-carbonyl)piperidin-3-yl]benzoic acid
5-fluoro-N-[1-(4-methylbenzoyl)piperidin-4-yl]quinazolin-4-amine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-{4-[4-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]phenyl}cyclopentanecarboxamide
N-[3-(2-methoxyphenoxy)propyl]-N-methylpyrrolidine-3-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
(5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
1-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-2-phenylethan-1-one
1-[3-(benzyloxy)azetidin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(morpholin-3-yl)acetamide
8-(6-carboxypyrazin-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}-3-methylbutan-1-one
N-{1-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
3-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
3-[2-(2,4-difluorophenyl)ethyl]-1-(prop-2-ene-1-sulfonyl)piperidine
N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
2-(1-methyl-1H-pyrrol-2-yl)-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-2-oxoacetamide
N-({7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
(4aS,8aR)-6-[(3,5-dichloropyridin-4-yl)methyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-(2-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
3-butyl-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-methylpiperazin-2-one
1-(5-fluoropyridin-3-yl)-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetic acid