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N-[(4-methoxypyridin-2-yl)methyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
1-(8-fluoroquinoline-2-carbonyl)-4-phenylpiperidin-4-ol
1-(4-methoxyphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]cyclopropane-1-carboxamide
1-methyl-4-{3-methyl-5-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl}piperidine
N-(1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
N-[2-(4-methoxyphenyl)ethyl]-1-methyl-N-(pyridin-2-ylmethyl)piperidine-2-carboxamide
4-(3,4-difluorobenzoyl)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N,N-dimethyl-3-({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}sulfamoyl)benzamide
2-(furan-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[benzyl(methyl)amino]-N-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-{3-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
1-methyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
1-(3-methylpyridin-4-yl)-4-[3-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepane
8-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}-1H-pyrazole
2-(oxolan-2-ylmethoxy)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
2-(dimethylamino)-2-(2-methylphenyl)-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}acetamide
5-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N,N-dimethyl-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine-1-sulfonamide
7-(cyclobutylmethyl)-2-[2-(pyrimidin-2-ylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-2-yl)methanol
methyl[3-(5-methylfuran-2-yl)butyl](pyrazin-2-ylmethyl)amine
3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
N-[(3R,4S)-4-cyclopropyl-1-(3-hydroxypropyl)pyrrolidin-3-yl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
5-[(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-(1-benzyl-1H-pyrazol-3-yl)-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
2-butanoyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-(2-methyl-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3R,4R)-1-(5-chloropyridin-2-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
N-benzyl-2-[4-(4-{[3-(pyridin-3-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
methyl (2S)-2-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]-2-phenylacetate
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
2-(2-ethylphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-(4-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-chloro-N-[2-(2-methoxy-5-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenoxy)ethyl]benzamide
ethyl 4-[1-(3-hydroxypyridine-2-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
11-[(cyclopropylmethyl)amino]-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
ethyl 1-benzyl-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{4-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]butyl}azepane
1-[2-({[(3-chlorophenyl)methyl]amino}methyl)-6-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
(2S,4R)-4-amino-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-N-ethylpyrrolidine-2-carboxamide
4-(3-phenylpropyl)-N-(1-propyl-1H-pyrazol-5-yl)-1,4-diazepane-1-carboxamide
5-[1-(2-methylpropyl)pyrrolidin-2-yl]thiophene-2-carboxamide