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7-(cyclobutylmethyl)-2-(3,6-dimethylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
2-amino-1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-methylpropan-1-one
3-[(3R,4S)-1-(2,5-dimethylfuran-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
(3R,4S)-3,4-dimethyl-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-ol
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
1-[2-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[3-(5-methylfuran-2-yl)butyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)propanamide
2-[5-(5-chloro-2-fluorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
7-(3-chlorophenyl)-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(pyrrolidin-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazole-5-carboxamide
5-cyclobutyl-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1,3,4-oxadiazol-2-amine
1-{1-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}piperidin-3-ol
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
4-[4-(4-chlorophenyl)butanoyl]morpholine-2-carboxamide
1-({5-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
4-{2-[(4-benzyl-5-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}morpholine
5-methoxy-3-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-indole-2-carboxamide
N-(2-methoxyethyl)-6-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(1S,5R)-6-(2-methoxyethyl)-3-(1-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-phenylpiperazin-1-yl)-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}propan-1-one
7-[(2-fluorophenyl)methyl]-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-ethyl-9-[(4-fluoro-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)-4H-chromen-4-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl][1-(4-methylpyridin-2-yl)propan-2-yl]amine
1-ethyl-N-[(4-fluorophenyl)methyl]-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2H-1,3-benzodioxol-4-ylmethyl)(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
2-(furan-2-yl)-N-(1-methyl-1H-1,3-benzodiazol-6-yl)azepane-1-carboxamide
(3R,4R)-1-(5-fluoro-3,8-dimethylquinolin-2-yl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-(morpholin-4-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}cyclopropane-1-carbonitrile
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
N-(adamantan-1-yl)-4-(4-methoxyphenyl)-3-oxopiperazine-1-carboxamide
4-(3-methoxypyrazin-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-cyclopentyl-4-oxo-4-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]butanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]butan-1-one
4-[5-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
3-{[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]sulfamoyl}-N-propylbenzamide
3-(3-acetyl-2-fluorophenyl)-N,N-dimethylbenzamide
N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-{1H-pyrrolo[2,3-b]pyridin-1-yl}acetamide
2-cyclopropyl-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
2-[4-(4-methylphenoxy)piperidin-1-yl]pyrazine
(2-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]morpholin-2-yl}ethyl)dimethylamine
2-(2-methoxyethoxy)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
2-amino-7-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-ethyl-3-(N-methylmethanesulfonamido)-N-{[4-(propan-2-yl)phenyl]methyl}propanamide
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one