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1-[2-(benzenesulfonyl)ethyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]azepan-2-one
2,6-dimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}quinoline-4-carboxamide
4-chloro-1-methyl-3-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-1H-indazole
N-(5-chloro-2-methoxyphenyl)-3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carboxamide
3-(2-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)(pyridin-3-ylmethyl)amine
8-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-N-(propan-2-yl)-1,3-benzoxazole-6-carboxamide
N-benzyl-N-(2-hydroxyethyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-(2-methoxyphenoxy)propanamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(1-phenoxypropan-2-yl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-(3-methylbutyl)-8-{[4-(methylsulfanyl)phenyl]methyl}-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-methoxy-2-methylbenzoyl)-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
5-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-2-ethylpyrimidine
2-[(4aR,7aS)-4-[2-(3,4-dimethylphenoxy)ethyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[3-(3-methylpyridin-4-yl)phenyl]acetamide
5-(pyridin-4-yl)-N-[1-(thiophen-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-({1-[(2,3-difluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)-3-ethylurea
methyl (2R,4S)-4-hydroxy-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-2-carboxylate
(1-{5-[(1-ethylpiperidin-4-yl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-yl)methanol
2-(3-fluoropyridin-4-yl)-5-(1H-imidazol-1-ylmethyl)pyridine
(1R,2R,4R)-N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-(carbamoylmethyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
3-methyl-7-(4-phenyl-1H-imidazole-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(2H-1,3-benzodioxol-5-yl)-N-cyclopentyl-N-{[3-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}acetamide
3-{[2-(2,4-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
propan-2-yl 4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxylate
(4aR,7aS)-1-benzyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-chloro-5-fluorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
2-(3-methoxypiperidine-1-carbonyl)-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
2-amino-4-[1-(2-methoxyethyl)piperidin-4-yl]-5-methyl-6-phenylpyridine-3-carbonitrile
4-methoxy-N-{[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
6-fluoro-4-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
1-methyl-N-(3-phenylpropyl)-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(4,4-difluoropiperidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
2-methyl-5-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-1,3,4-thiadiazole
4-[(1-{[1-(2-methylpyrimidin-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
1-(2-{[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]amino}ethyl)piperidin-3-ol
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(pyridin-4-yl)pyrimidine
2-{[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]methyl}-6-methoxyphenol
4-benzyl-3-ethyl-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1,4-diazepan-5-one
6-methoxy-3-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}quinolin-2-ol
(2R,6S)-2,6-dimethyl-4-[5-(pyrrolidin-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]morpholine