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1-[4-(furan-2-ylmethyl)piperazin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
(1R,3S)-3-[(2-methoxyethyl)(pyridin-3-ylmethyl)carbamoyl]cyclopentane-1-carboxylic acid
6-(propan-2-yl)-N-[1-(pyridin-4-yl)propyl]pyrimidin-4-amine
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
3-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]urea
1-{7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-phenylethan-1-one
N,N-dimethyl-1-(prop-2-en-1-yl)-5-({[2-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(5-methyl-1H-pyrazol-1-yl)-1-[5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
N-ethyl-2,6-dihydroxy-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
[3-(cyclopropylmethyl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]methanol
3-(1H-1,3-benzodiazol-1-yl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}propanamide
2-(4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenol
N-{2-[bis(propan-2-yl)amino]ethyl}-1-(carbamoylmethyl)piperidine-3-carboxamide
N-[2-(azepan-1-yl)ethyl]-4-methanesulfonyl-N-(propan-2-yl)benzamide
(2S,3R)-2-({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)-3-hydroxybutanamide
5-methyl-5-[1-(4-phenyl-1H-imidazole-5-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[(2-ethoxyphenyl)methyl]-N-ethyl-4-(1H-1,2,4-triazol-1-yl)butanamide
2-(3-chloro-4-hydroxyphenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-2-methyl-3-(1H-pyrazol-1-yl)propanamide
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl][(2-methoxyphenyl)methyl]methylamine
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}benzamide
(2S,4R)-1-(1H-imidazol-2-ylmethyl)-4-(5-methoxyfuran-2-amido)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-benzyl-8-(1H-indol-2-ylmethyl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}benzonitrile
1-{3-[4-(3-methylphenyl)piperazin-1-yl]propanamido}cyclopentane-1-carboxamide
N-(furan-2-ylmethyl)-5-{1-[(2-hydroxyphenyl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(pyridin-4-yl)propanamide
N-(pyrimidin-4-ylmethyl)-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(3R,4R)-4-amino-1-[1-(4-chlorophenyl)cyclohexanecarbonyl]piperidin-3-ol
methyl 5-methyl-4-{2-[1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-imidazol-4-yl}furan-2-carboxylate
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
5-tert-butyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3,4-oxadiazol-2-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]acetamide
[2-(1H-1,3-benzodiazol-2-yl)ethyl](5-methylhex-5-en-2-yl)amine
N-cyclopropyl-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}-3-phenyl-1H-pyrazole-5-carboxamide
(4aR,6R,8aS)-2-[(4,5-dimethylfuran-2-yl)methyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
(2S)-2-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamido]-3-phenylpropanamide
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-5,6,7,8-tetrahydroquinazolin-2-amine
2-methyl-N-{3-[methyl(phenyl)amino]propyl}imidazo[1,2-a]pyridine-6-carboxamide
methyl 2-{[5-acetamido-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazol-7-yl]formamido}-4-(methylsulfanyl)butanoate
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-(5-fluoro-2-methylphenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
2-(2-acetyl-1H-1,3-benzodiazol-1-yl)-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]pyrrolidine-1-carboxamide
2-{8-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
1-[(2-ethylpyrimidin-4-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-[4-(piperidin-1-ylmethyl)benzoyl]azetidine-2-carboxylic acid
methyl 4-[(7-oxo-4-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,4-diazepan-1-yl)methyl]benzoate