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N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-(ethylamino)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}pyrimidine-5-carboxamide
4-{[7-acetyl-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-1-propylpyrrolidin-2-one
3-(1H-imidazol-1-yl)-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazine
4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(methoxymethyl)-6-(3-methyl-3-phenylpiperidine-1-carbonyl)pyridine
2-(3-{[propyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(propan-2-yloxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4-sulfamoylphenyl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(cyclohexylmethyl)-2-(2,2-dimethylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
3-({2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-cyclopentyl-9-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[(4-methyl-1H-imidazol-5-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
8-(butan-2-yl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(benzylsulfamoyl)(2-methylpropyl)(thiophen-3-ylmethyl)amine
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[3-(morpholin-4-yl)propyl]propanamide
(3S,4S)-4-({[2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidin-4-yl]amino}methyl)piperidin-3-ol
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-3-(piperidin-3-yl)benzamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
4-(1H-imidazole-5-carbonyl)-2-[(4-methoxyphenyl)methyl]morpholine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(5-ethylfuran-2-yl)methyl](2-methoxyethyl)amine
N-[(2,3-dimethoxyphenyl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}bis(1,3-oxazol-4-ylmethyl)amine
1-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)ethan-1-one
2-(1H-indol-3-yl)-N-methyl-N-(oxan-2-ylmethyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-cyclopentyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methylpyrimidin-2-amine
1-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-yl}piperidin-4-ol
N-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-4-[(4-fluorophenyl)methyl]piperazine-1-carboxamide
3-{[2-(aminomethyl)morpholin-4-yl]methyl}-6-methoxyquinolin-2-ol
3-chloro-N-cyclopentyl-4-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}benzamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(oxan-4-yl)amino]methyl}piperidin-2-one
4-{4-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]piperazin-1-yl}-2-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[(ethylsulfanyl)methyl]-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[4-(4-{[(3-fluoro-4-methylphenyl)methyl]amino}piperidin-1-yl)phenyl]-2-(4-methoxyphenyl)acetamide
(2S,4S)-N-[2-(4-fluorophenyl)ethyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
2-(3,4-dichlorophenyl)-4-{2-methylthieno[2,3-d]pyrimidin-4-yl}morpholine
6-(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(4-fluorophenyl)-4-[(3-{2-[1-(furan-2-carbonyl)piperidin-2-yl]ethoxy}-4-methoxyphenyl)methyl]piperazine
3-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
3-{[4-(2,2-dimethylpropanoyl)piperazin-1-yl]methyl}-N-(1-methyl-1H-1,2,4-triazol-3-yl)benzamide
5-ethyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-(oxolan-2-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]thiophene-2-carboxamide
{4-[(3-methoxyphenyl)methyl]piperidin-4-yl}methanol
2-[(4aS,8aR)-2-oxo-1-propyl-decahydro-1,6-naphthyridine-6-carbonyl]benzonitrile
2-[4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
1-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-3-phenoxypropan-1-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
(4aS,8aR)-6-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one