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({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[2-(1,3-thiazol-4-yl)ethyl]amine
13-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4,6-dimethyl-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-4-yl}propanamide
8-methoxy-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-cyclopropyl-N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1H-pyrazole-5-carboxamide
N-[(2-ethoxyphenyl)methyl]-N-ethyl-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-[2-(morpholin-4-yl)ethyl]-4-{4-[4-(pyrimidin-2-yl)piperazin-1-yl]piperidin-1-yl}benzamide
9-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(morpholin-4-yl)ethyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-methyl-5-(piperidin-4-yl)-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}imidazolidine-2,4-dione
N-cyclopropyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}propanamide
9-[(3,5-dimethoxyphenyl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
(3aR,6aS)-5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
(2S,4S)-N-ethyl-4-[3-(ethylsulfanyl)propanamido]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
methyl 4-{[(2S,4R)-2-{[2-(3-chlorophenyl)ethyl]carbamoyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidin-1-yl]methyl}benzoate
N-{1-[1-(2-phenoxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N-({1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
(3aS,6aS)-2-(furan-2-carbonyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1H-indol-4-ylmethyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(2-methylpropyl)acetamide
N-[(3S,4R)-1-(5-fluoropyrimidin-2-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
(2S)-1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}pyrrolidine-2-carboxamide
N-({1-[2-(carbamoylamino)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-4-methylbenzamide
1-(cyclohex-3-en-1-ylmethyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
1-{2-[methyl({[3-(2-methylphenyl)phenyl]methyl})amino]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(4-carbamoyl-1,3-thiazol-2-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-[2-(dimethylamino)ethyl]-8-[4-(methylsulfanyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(3-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}propanamido)acetic acid
5-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,2-dimethyl-1H-imidazole
(3S,4S)-4-cyclopropyl-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidine-3-carboxylic acid
1-cyclopropanecarbonyl-N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)piperidine-4-carboxamide
1-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-one
4-hydroxy-1-(4-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxylic acid
1-(3-methoxyphenyl)-3-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}urea
1-benzyl-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-(propan-2-yl)-5-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1,2,4-oxadiazole
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
(1R,9aR)-1-({[2-(pyrrolidine-1-sulfonyl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
ethyl 1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxylate
8-[(2,3-difluoro-4-methylphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-[3-chloro-4-(propan-2-yloxy)phenyl]-1-(oxan-4-ylmethyl)urea
N'-(adamantan-1-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanediamide
3-(3,4-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
4-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}benzonitrile
2-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
methyl 3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-4-hydroxy-2-methylpyrimidine-5-carboxamide
3-butyl-4-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1-methylpiperazin-2-one