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7-(1-ethylpiperidine-4-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-amino-4-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-5-carboxamide
4-{1-ethyl-5-[(2-oxo-1,2-dihydropyridin-1-yl)methyl]-1H-1,2,4-triazol-3-yl}benzamide
1-methyl-6-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1H-indole
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
6-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
(3aS,6aS)-2-(ethanesulfonyl)-5-(1H-imidazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-2-(methylsulfanyl)pyrimidine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(2,4-difluorophenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
2-[(dimethylamino)methyl]-4-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-imidazol-2-yl}phenol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(dicyclopropylmethyl)-1,3-oxazole-4-carboxamide
1-propyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}piperidin-4-amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-(6-chloropyridin-3-yl)-3-[(1-ethylpyrrolidin-3-yl)methyl]urea
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
N-[2-(pyridin-3-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-[2-(3-ethenylphenyl)-1H-imidazol-1-yl]propan-1-ol
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-{[(4-methylphenyl)methyl]amino}-N-[2-(2-oxopyrrolidin-1-yl)ethyl]benzamide
1-[(3-methylquinoxalin-2-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}acetamide
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-{[2-(2-hydroxyethoxy)phenyl]methyl}-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-tert-butyl-2,6-dimethyl-N-(thiophen-3-ylmethyl)pyrimidine-4-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
N-(pentan-3-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
3-(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)benzoic acid
1-(3,5-difluorophenyl)-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2S,4S)-4-[(adamantan-2-yl)amino]-1-[(4-chlorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3-oxazolidin-2-one
5-acetyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]thiophene-3-carboxamide
methyl[(3-methyl-1H-indol-2-yl)methyl]{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
2-methyl-6-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
2-{3-[3-(pyridin-2-yl)azetidine-1-carbonyl]piperidin-1-yl}pyridine
2-(2,3-dimethoxy-5-methylphenyl)-6-fluorobenzamide
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
N,N-dimethyl-7-(1-methyl-1H-imidazole-5-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{[3-(dimethyl-1,3-thiazol-5-yl)phenyl]methyl}morpholine
(3R,4R)-4-cyclobutyl-3-methyl-1-(thiophene-2-carbonyl)piperidin-4-ol
2-amino-6-(pyridine-4-carbonyl)-4-(thiophen-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(4aS,7aR)-1-(2-hydroxybenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-({4-methyl-5-[1-(propan-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-(4-hydroxy-3-methoxyphenyl)-4-(2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]quinoxaline
4-[1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
(3R,4R)-3,4-dimethyl-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-ol