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(3aR,6aR)-2-methanesulfonyl-5-[2-(2-methylphenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,3R)-N1-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
methyl 4-({[2-(5-oxo-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}pyrrolidin-2-yl)ethyl]amino}methyl)benzoate
(4aR,7aS)-1-acetyl-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3-{2-[1-(3-chlorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](furan-2-ylmethyl)(3-methylbutan-2-yl)amine
N-[4-(1-methyl-1H-imidazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
1-(3-hydroxypropyl)-4-(1H-indol-2-ylmethyl)-1,4-diazepan-6-ol
5-methyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-(5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
2-(dimethylamino)-8-(1H-imidazol-4-ylmethyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-methyl-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
1-{[3-(2-aminoethyl)phenyl]methyl}-1,4-diazepane-6-carboxylic acid
N-methyl-N-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}thian-4-amine
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]thiophene-2-carboxamide
1-[(5-{[3-(2-aminoethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
1-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
1-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1H-indazole
N-[(3S)-2-oxoazepan-3-yl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-ethoxyethan-1-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}imidazo[1,2-a]pyrimidine-2-carboxamide
methyl 3-methyl-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N2,N4,N4,5-tetramethyl-N2-(1H-pyrazol-5-ylmethyl)pyrimidine-2,4-diamine
(2S,4S)-4-amino-1-(4-methoxycyclohexanecarbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-3-(pyrrolidin-1-yl)piperidine
3-methoxy-1-{4-[4-(thiomorpholine-4-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
3-(2-fluorophenyl)-3-phenyl-N-(pyridin-4-ylmethyl)propanamide
1'-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
6-(2,4-dimethoxyphenyl)-N4-methylpyrimidine-2,4-diamine
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-2-(1-tert-butyl-1H-pyrazol-4-yl)quinoline
2-{[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]methyl}-6-chloro-1,4-dihydroquinolin-4-one
N-[1-(1H-indol-2-yl)ethyl]-N,5-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N,1-dimethyl-N-[2-(4-methylpiperidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(morpholin-2-yl)acetamide
4-phenyl-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butane-1,2-dione
N,N-dimethyl-5-(5-phenyl-1,2-oxazole-4-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
5-methoxy-2-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
4-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
methyl (2S,4S)-1-methyl-4-(1-phenyl-1H-1,2,3-triazole-5-amido)pyrrolidine-2-carboxylate
4-[(6-chloropyridin-2-yl)methyl]-2-(3,4-dichlorophenyl)morpholine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
N-benzyl-N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-phenyl-1-[1-(pyridin-4-ylmethyl)piperidin-3-yl]ethan-1-one
8-(3-hydroxypropanoyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-(2-cyclopropylacetyl)-4-(pyrimidin-2-ylmethyl)-1,4-diazepane-6-carboxylic acid