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5-(4-ethylpiperazin-1-yl)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}cyclopropanecarboxamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-[2-(ethylsulfanyl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(3-chlorophenyl)methyl]-3-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]propanamide
1-cyclohexyl-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
6-methyl-2-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-1,2-dihydropyridine-4-carboxamide
N-(2-oxoazepan-3-yl)-4-(1H-pyrazol-3-yl)benzamide
2-[5-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]acetic acid
N-ethyl-N-(oxan-4-ylmethyl)-3-propyl-1H-pyrazole-5-carboxamide
2-amino-4-(4-methoxynaphthalen-1-yl)-6-methyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-cyano-N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-1-methyl-1H-pyrrole-2-carboxamide
2-(1-methyl-1H-pyrazol-4-yl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridine
3-(5-methyl-1H-indol-3-yl)-5-(morpholine-4-sulfonyl)benzoic acid
[(2-ethylpyrimidin-4-yl)methyl](methyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
5-benzyl-5-(1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[4-(3-propanoylphenyl)phenyl]acetamide
N-[3-(4-chlorophenyl)propyl]-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
2-amino-4-[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
7-(1-benzothiophen-3-yl)-4-cyclopropanecarbonyl-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 4-[2-(2-phenylethyl)morpholine-4-carbonyl]benzoate
3-(2-methoxyethyl)-1-(4-methyl-2-oxo-2H-chromen-7-yl)-3-[(5-methylthiophen-2-yl)methyl]urea
2-methyl-5-{3-methyl-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}pyrazine
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-(3-methylthiophene-2-carbonyl)piperidine
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-2-(1,2-oxazolidin-2-yl)pyridine
5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-(2-phenylethyl)-1,3-benzoxazole
N-benzyl-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
2-ethyl-9-[2-(methylsulfanyl)acetyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
5-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridin-4-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-ethyl-N-methyl-3-(pyrrolidine-1-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(6-chloropyridin-2-yl)methyl]-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[methyl(prop-2-en-1-yl)amino]methyl}piperidin-2-one
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-6-oxo-1-propylpiperidine-3-carboxamide
2-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}benzoic acid
2-(2,3-dimethoxyphenyl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N,5-dimethyl-6-(piperidine-1-carbonyl)-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
2-amino-1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpropan-1-one
N-({3,5-dimethoxy-4-[2-(1-methylpyrrolidin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]cyclobutanecarboxamide
N-{[2-(2,5-dimethoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}cyclopentanamine
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]propanamide
N-[(5-methylpyrazin-2-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
(1R,5R)-6-benzyl-3-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-cyclopropyl-3-(3-fluorophenyl)-N-[(3-hydroxyphenyl)methyl]-1H-pyrazole-4-carboxamide
4-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(5-methylpyridin-3-yl)benzamide
1-(4-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one