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1-(2-chlorophenyl)-4-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperazin-2-one
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)thiophene-3-carboxamide
2-amino-4-ethyl-6-(3-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl 8-(2,3-dihydro-1H-inden-2-yl)-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(2R)-2-methylpyrrolidine-2-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-[(2-ethyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-2-{imidazo[1,2-a]pyridin-3-yl}acetamide
2-amino-6-{4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}pyrimidin-4-ol
N-[2-(3-methylpiperidin-1-yl)ethyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carbonitrile
4-[2-(3-methoxyphenoxy)ethyl]-N,N-dimethylbenzamide
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopentanecarboxamide
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-(pyrrolidin-1-yl)pyrazine
N-[4-(propan-2-yl)phenyl]-1-(1,3-thiazole-4-carbonyl)piperidin-3-amine
N-methyl-1-(propan-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]piperidine-4-carboxamide
1-[4-(dimethylamino)azepan-1-yl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propan-1-one
1-(4-methyl-1,3-thiazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-(1,4-oxazepan-6-ylmethyl)-3-[4-(pyridin-2-ylmethoxy)phenyl]urea
2-cyclopropyl-8-(2-phenoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-methoxy-2-methylphenyl)methyl]pyrrolidine-3-carboxylic acid
1-(3-methanesulfonamidophenyl)-3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
4-ethyl-3-{1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-(methylsulfanyl)acetamide
4-{[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzoic acid
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrrolidine-3-carboxamide
2-(dimethylamino)-N-[2-(pyridin-3-yloxy)propyl]-2,3-dihydro-1H-indene-2-carboxamide
5-butyl-6-methyl-N4-(1,2-oxazol-3-ylmethyl)pyrimidine-2,4-diamine
(1S,5R)-3-benzyl-6-(4-fluoro-2-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(2-fluorophenyl)formamido]-N-[1-(thiophen-2-yl)propyl]propanamide
1-[(4aR,8aR)-4a-hydroxy-7-(thiophen-3-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-[2-(furan-2-yl)ethyl]-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
4,5-dimethyl 1-[(3S,5S)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5-[(quinolin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
2-{3-[1-(but-3-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyridine
2-{methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-4-[(2-methylpropanamido)methyl]benzamide
N-(2-phenylethyl)-1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}propan-1-one
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-phenyl-1,3-oxazole
N-[(6-chloropyridin-3-yl)methyl]-7-fluoro-N,2-dimethylquinoline-4-carboxamide
5-ethyl-2,3-dimethyl-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4,6-dimethyl-2H-pyran-2-one
N-(2-methoxyethyl)-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(propan-2-yl)propanamide
2-(dimethylamino)-N-ethyl-2-(3-methylphenyl)-N-(pyridin-4-ylmethyl)acetamide
6-methyl-2-(2-{4-[2-(3-methylphenyl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
4-(2-{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}ethyl)phenol
1-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
3-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
(2S,4S)-4-amino-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide