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ethyl 5-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-fluoro-N-(2-{[5-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]formamido}ethyl)benzamide
1-(4-methylphenyl)-4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazin-2-one
2-ethyl-N-(1-methoxypropan-2-yl)-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-{3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]morpholin-4-yl}propan-1-one
1-{[4-(dimethylamino)phenyl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-{4-[3-(methylsulfanyl)phenyl]phenyl}acetamide
1-(but-3-enoyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
3-cyclopentyl-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
7-[(3,4-difluorophenyl)methyl]-2-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(3R)-1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-3,4,4-trimethylpyrrolidin-3-ol
(2S)-1-(1-{3-[3-(trifluoromethyl)benzamido]phenyl}piperidin-4-yl)pyrrolidine-2-carboxamide
2-(2-butoxy-4-fluorophenyl)-2-(dimethylamino)acetic acid
3-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
(2S,4R)-4-amino-N,N-diethyl-1-[2-(4-methoxyphenoxy)acetyl]pyrrolidine-2-carboxamide
3-fluoro-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-cyclopentanecarbonyl-N-{[4-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxamide
1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N,1-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-3-yl)acetamide
N-ethyl-4-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]piperidine-1-carboxamide
N-[(1R)-1-(4-methoxyphenyl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
3-(2,3-dimethoxyphenyl)-1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}pyrrolidine
3-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
5-[3-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
(4aR,8aR)-4-[(3-fluoro-2-methoxyphenyl)methyl]-octahydro-2H-1,4-benzoxazine
N-(2,5-dimethylphenyl)-N'-methyl-N'-[1-(pyrimidin-4-yl)ethyl]propanediamide
1-[2-methoxy-5-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
1-[2-(3-methoxyphenyl)piperidin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
1,4-dimethyl-N-[4-(pentyloxy)phenyl]-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
5-(1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1H-imidazol-2-yl)-2-(pyridin-2-yl)pyrimidine
2-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-benzofuran-7-carboxamide
[(1-{[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
3-(2,4-dimethoxybenzoyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine
(4S)-3-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
5-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-phenylethane-1,2-dione
1-[(4aR,8aR)-4a-hydroxy-7-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
N,N-diethyl-5-[1-(3-methylfuran-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(1R,3S,5S)-8-(6-ethyl-2-methylquinoline-4-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
2-{2-[3-(1H-pyrazol-3-yl)phenyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
1-(1-benzofuran-3-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
methyl (2S)-1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl}pyrrolidine-2-carboxylate
2-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N,4,6-trimethyl-2-oxo-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
3-(1H-pyrazol-1-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-chloro-4-{[(oxan-4-yl)carbamoyl]amino}benzamide