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2,5-dimethyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
5-methyl-N-[2-(morpholin-4-yl)ethyl]-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-1,2-oxazinane
2-cyclopropyl-1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}amine
1-[1-(6-cyanopyridin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
1-(oxan-4-yl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(1S,3R)-3-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamido]-N-phenylcyclopentane-1-carboxamide
1-(2-{1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
2-(1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
4,5-dimethyl-2-[5-(oxolane-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1H-1,3-benzodiazole
7-[(3,4-difluorophenyl)methyl]-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepane
4-[3-(morpholine-4-carbonyl)piperidine-1-carbonyl]benzene-1-sulfonamide
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(morpholin-4-yl)ethan-1-one
7,7-dimethyl-2-[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}pent-4-en-1-one
5-chloro-N-(1-cycloheptylpiperidin-3-yl)-2-fluorobenzamide
2-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
methyl[(1-methylpiperidin-4-yl)methyl]{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
2-acetyl-8-(oxan-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(piperidin-4-ylmethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[(1S,5R)-6-(7-chloro-2-methylquinoline-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-{4-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]phenyl}acetic acid
3-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}-N-phenylpropanamide
5-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]-3-propyl-1,2,4-oxadiazole
[(2S,4R)-4-(dimethylamino)-1-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-2-yl]methanol
N-{[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]methyl}-1H-indole-5-carboxamide
N-(1-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
2-methyl-6-({4-[4-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-{6-[4-(2-hydroxypropan-2-yl)piperidin-1-yl]pyridin-3-yl}ethan-1-one
4-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-N-(trimethyl-1H-pyrazol-4-yl)benzamide
4-chloro-N-methyl-3-{[methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})carbamoyl]amino}benzamide
(2S,4S)-4-amino-1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-(1-methyl-1H-pyrazol-3-yl)acetamide
3-(4-fluorophenyl)-3-phenyl-N-(1H-1,2,4-triazol-5-ylmethyl)propanamide
ethyl 3-{[5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazol-4-yl]formamido}propanoate
1-(3-methanesulfonylbenzoyl)-2-(pyrrolidine-1-carbonyl)piperazine
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-3,4-dihydroquinazolin-4-one
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[(3-propyl-1,2-oxazol-5-yl)methyl]urea
3-(2-benzylphenyl)-1-[3-(4-methylpiperazin-1-yl)butyl]urea
3-(2-ethylbutyl)-8-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl[(2-propylpyrimidin-5-yl)methyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
(1R,5S,6S)-6-{[4-(2-ethylphenyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]-5-methoxyphenol
3-(1,3-benzothiazol-2-yl)-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]propanamide
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-5-fluoroquinazolin-4-amine