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2-{2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-4,6-dimethylpyridine-3-carbonitrile
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1H-indole-3-carboxamide
3-(4-fluorophenyl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3-phenylpropanamide
4-{4-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-[3,5-dimethyl-4-(pyridin-3-yl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
N-[(2S)-2,3-dihydroxypropyl]-5-methyl-1,3-diphenyl-1H-pyrazole-4-carboxamide
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenol
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
2-(2-aminoethyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]quinazolin-4-amine
1-cyclopentanecarbonyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
N-[(3R,4S)-1-[(6-methylpyridin-2-yl)methyl]-4-propylpyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-3-(thiophen-3-yl)-1H-pyrazole
7-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[4-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
N,N-diethyl-3-{[(thiophen-3-ylmethyl)amino]methyl}pyridin-2-amine
(3S,4R)-1-(carboxymethyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-methoxy-5-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}pyridine
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-N-[(3,4,5-trifluorophenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methoxy-8-(2-phenylethyl)-1,8-diazaspiro[4.5]decan-2-one
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
4-(cyclohex-3-en-1-ylmethyl)-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5,6-dihydrophenanthridin-6-one
2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propane-1,3-diol
5-{[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-[(2-amino-6-{methyl[(3-methylthiophen-2-yl)methyl]amino}pyrimidin-4-yl)amino]ethan-1-ol
4-(2-methyl-1,4-oxazepane-4-carbonyl)-2-(pyridin-4-yl)quinoline
3-(azocane-1-carbonyl)-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
7-(5-methyl-1H-indol-3-yl)-1,2-dihydroisoquinolin-1-one
4-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-1-(1H-indazol-6-yl)piperazin-2-one
2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]-N-(1,2-oxazol-5-ylmethyl)acetamide
8-(3-fluoropyridin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-{[4-(furan-2-yl)butan-2-yl]amino}pyrimidin-4-yl)piperidin-4-ol
2-[2-(4-benzyl-1,4-diazepan-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
(2E)-N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3,4-dimethoxyphenyl)prop-2-enamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-(pyridin-3-yl)propanamide
N-(2-phenoxyethyl)-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
1-(1H-imidazol-4-ylmethyl)-3-[2-(3-methoxyphenyl)ethyl]piperidine
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-chloro-4-{1-[2-(2-hydroxyethoxy)ethyl]-4-phenyl-1H-imidazol-5-yl}phenol
4-methyl-2-phenyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
6-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-benzothiazole
(4aS,8aR)-6-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-[2-(4-methanesulfonylphenyl)ethyl]-3,5-dimethyl-1H-pyrazole