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3-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}-N-(1,2,4-thiadiazol-5-yl)benzamide
ethyl 1-[2-(2-oxopyrrolidin-1-yl)acetyl]-4-(2-phenylethyl)piperidine-4-carboxylate
(1S,6R)-3-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(morpholin-4-yl)ethan-1-one
(1R,7S)-3-cycloheptyl-N-ethyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
methyl 1-{2-hydroxy-3-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}piperidine-4-carboxylate
2-amino-N-({1-[(2E)-2-methylpent-2-en-1-yl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
[6-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)pyridin-2-yl]methanol
N-[3-(methylamino)propyl]-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
methyl 4-({1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}carbamoyl)butanoate
3-{6-ethyl-4-oxo-5-phenyl-3H,4H-thieno[2,3-d]pyrimidin-3-yl}-1-methylpyrrolidin-2-one
8-[2-(benzylamino)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(4-fluorophenoxy)pyridin-3-yl]-7-methyl-2,7-diazaspiro[4.4]nonane-2-carboxamide
4-{2-[4-(dimethylamino)phenyl]acetyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
N-cyclohexyl-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(pyridin-3-ylmethyl)acetamide
2-({4-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]phenyl}(methyl)amino)ethan-1-ol
4-{[(butan-2-yl)(cyclopentyl)amino]methyl}-N-methylbenzene-1-sulfonamide
1-[2-(4-methoxyphenyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
8-[(4-hydroxyphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2-methoxyacetyl)-N-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-1,4-diazepane-1-carboxamide
[4-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-1,4-oxazepan-6-yl]methanol
N-{4-oxo-4-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butyl}acetamide
N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}piperidin-2-one
N-ethyl-3-methyl-N-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}aniline
5-methyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-1,3-oxazole-4-carboxamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine-4-carboxylate
N-cyclopropyl-4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(1H-indol-5-ylmethyl)benzamide
3-{2-oxo-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}-1,3-oxazolidin-2-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methanol
(1R,5S,6R)-3-[(1S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N-(pyridin-3-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
8-[(3-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
5-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
2-(3-{[(1R,5S,8R)-8-(dimethylamino)-3-azabicyclo[3.2.1]octan-3-yl]methyl}phenoxy)acetamide
(1S,5R)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(3aR,6aR)-2-(2-methoxyacetyl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
6-[2-(azocan-1-yl)-2-oxoethyl]-5,6-dihydro-1,6-naphthyridin-5-one
(2S,4R)-4-amino-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrrolidine-2-carboxamide
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
2-acetyl-8-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-(4-fluorophenyl)propyl]-3-[4-(morpholin-4-ylmethyl)phenyl]urea
2-methyl-5-{[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrazine
1'-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
3-benzoyl-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidine