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N-[1-(4-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethyl]acetamide
2-[(1S,5R)-6-(3-cyanobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
3-(1-butyl-1H-imidazol-2-yl)-N,N-dimethylpiperidine-1-sulfonamide
4-[(3-fluorophenyl)methyl]-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
3-methyl-6-[5-(2-methylbutan-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-methylphenyl)ethan-1-one
N-[2-(1-hydroxycyclopentyl)ethyl]-2-[(3-methoxyphenyl)amino]butanamide
5-[(2S)-2,3-dihydro-1H-indole-2-carbonyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methylbenzamide
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-(propane-1-sulfonyl)piperidine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(3-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
7-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-[4-(hydroxymethyl)piperidin-1-yl]-2-[4-(propan-2-yloxy)phenyl]acetic acid
3-[4-(4-methylphenyl)phenyl]-1-(morpholin-2-ylmethyl)urea
N-[2-(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
N-benzyl-3-methoxy-N-(prop-2-en-1-yl)pyridine-2-carboxamide
2-(3-acetyl-1H-indol-1-yl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}butanamide
(1R,2S)-1-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)-2,3-dihydro-1H-inden-2-ol
2-[benzyl(methyl)amino]-N-[(3S)-2-oxoazepan-3-yl]-2,3-dihydro-1H-indene-2-carboxamide
N3-[(2,6-difluoro-3-methoxyphenyl)methyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
2-({4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)benzonitrile
1-[1-(4-fluorobenzoyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
9-methyl-3-[4-(2-phenylpyrimidin-4-yl)piperidine-1-carbonyl]-9H-carbazole
2-(4-fluorophenyl)-N-[2-(morpholin-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
methyl({[4-(methylsulfanyl)phenyl]methyl})[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
ethyl 4-[(2-chlorophenyl)methyl]-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]acetamide
N-methyl-5-oxo-N-(1H-pyrazol-3-ylmethyl)-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
methyl 2-{2-oxo-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazin-1-yl}acetate
methyl (2S)-1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-yl]pyrrolidine-2-carboxylate
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-3-carbonyl)piperidine
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[3-(oxolan-2-yl)propyl]amine
(2R,6R)-11-methoxy-4-(pyridin-3-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(2-{[(2-cyclopropylphenyl)carbamoyl]amino}ethyl)acetamide
2-{6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}-1-methyl-1H-1,3-benzodiazole
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[3-(2-hydroxyethoxy)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
4-{1-[2-(2-chlorophenyl)ethyl]-1H-imidazol-2-yl}-3,5-dimethyl-1,2-oxazole
2-amino-6-(3-methoxyphenyl)-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
2-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-N-(propan-2-yl)acetamide
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-({3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
3-[(cyclopropylamino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-(cyclopropylmethyl)-4-(1H-imidazol-2-ylmethyl)-1,4-diazepane-6-carboxylic acid
N-(5-methyl-1,2-oxazol-3-yl)-2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]acetamide
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-2-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](1H-indol-3-ylmethyl)methylamine
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide