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{3-[(3-chlorophenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl}methanol
4-{4-[(2-oxopiperidin-3-yl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
N3-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-N1,N1-dimethylpiperidine-1,3-dicarboxamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(3-methoxyphenyl)methyl]piperidine
3-(methylsulfanyl)-N-(quinolin-2-ylmethyl)propanamide
4-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
3-(1-methyl-1H-pyrrol-2-yl)-5-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1H-pyrazole
2-butyl-4-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2,3-dihydro-1-benzofuran-7-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-3-(2-methyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
3-[(3R,4S)-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[2-(2-methoxyethoxy)phenyl]-2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
methyl (2S,4R)-1-{[5-(2-cyanophenyl)furan-2-yl]methyl}-4-(dimethylamino)pyrrolidine-2-carboxylate
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
2-methoxy-1-[1'-(quinolin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
4-ethyl-2-methyl-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-ethyl-N-(2-phenylethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-propyl-5-[4-(pyridin-2-ylmethyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(isoquinolin-5-ylmethyl)piperidin-4-yl]propanamide
8-(4-methoxybutan-2-yl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
2-[(4-cyclopentylpyrimidin-2-yl)amino]-N-(propan-2-yl)acetamide
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(pyrazin-2-yl)propanamide
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N,1-dimethyl-5-phenyl-1H-pyrrole-2-carboxamide
6-ethyl-N-[3-(4-fluorophenyl)propyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
6-methyl-2-[2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-3,4-dihydropyrimidin-4-one
(1S,5R)-6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-(4-fluorobenzoyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]benzamide
methyl (1R,3S,3aR,6aS)-3-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
6-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2-(pyridin-3-yl)pyrimidin-4-amine
(1r,4r)-4-{[2-(4-acetamidophenyl)-1H-imidazol-1-yl]methyl}cyclohexane-1-carboxylic acid
2-{4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]morpholin-3-yl}acetic acid
6-[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]quinoline
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
2-{4-[(2-chlorophenyl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
methyl 6-{[methyl(thiophen-3-ylmethyl)amino]methyl}-3-(1-phenylcyclopropaneamido)thieno[2,3-b]pyridine-2-carboxylate
4-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
2-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]-1H-1,3-benzodiazole
4-chloro-1,5-dimethyl-N-{2-[methyl(phenyl)amino]propyl}-1H-pyrazole-3-carboxamide
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-acetyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}benzamide
1-[(5-acetylthiophen-3-yl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(1-methyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aS,8aS)-2-cyclobutanecarbonyl-7-(5-ethyl-1H-pyrrole-2-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol