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8-(3-fluoro-2-methoxybenzoyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(1-benzyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-(trifluoromethyl)morpholine
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-[(2-methyl-1,3-oxazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-({[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]carbamoyl}methyl)piperidine-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[2-(2-oxopyrrolidin-1-yl)ethyl]pyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide
N-{[3-(2-fluoro-6-methoxyphenyl)phenyl]methyl}cyclopropanamine
({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
N-(furan-2-ylmethyl)-N-methyl-7-[(1-methyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-benzyl-4-[2-(2-cyclopropyl-1H-imidazol-1-yl)ethyl]piperazine
1'-[5-(methoxymethyl)thiophene-2-carbonyl]spiro[indene-1,4'-piperidine]
N-(3-carbamoylphenyl)-3-[(diethylamino)methyl]benzamide
6-methyl-N4-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)pyrimidine-2,4-diamine
5-{2-[5-(1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
N-(furan-2-ylmethyl)-2-(morpholin-4-yl)benzamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoic acid
methyl 1-{[4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(methoxymethyl)piperidine
1-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
2-{3-[3-(2-methylpyridin-4-yl)phenyl]-1H-pyrazol-1-yl}-N-(pyrazin-2-yl)acetamide
3-{[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
[(3R,4R)-1-(2-chlorobenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl})amine
N-[2-(azepan-1-yl)ethyl]-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-ethylacetamide
5-(3-methyl-3-phenylpiperidine-1-carbonyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
11-{[(5-methylpyrazin-2-yl)methyl]amino}-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(4aS,8aR)-6-[(2-fluorophenyl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
2-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
5-(pyrrolidin-1-ylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]furan-2-carboxamide
3-(5-{[cyclopropyl({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}thiophen-2-yl)prop-2-yn-1-ol
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
1-{5-[2-(3-phenylpropyl)morpholine-4-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
ethyl 1-[(2-methoxyphenyl)methyl]-1H-imidazole-2-carboxylate
N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
4-fluorophenyl (7S,9aR)-7-[(2S)-butan-2-yl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-[1-(propan-2-yl)piperidine-3-carbonyl]-4-(1H-pyrrole-2-carbonyl)piperazine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-methyl-1,3-benzoxazole-6-carboxamide
2-[(2-hydroxyethyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]ethan-1-ol
2-[3-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}methyl)phenyl]-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
1-ethyl-3-[3-(pyridin-3-yl)propyl]-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-methylphenoxymethyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
2-(2-oxopyrrolidin-1-yl)-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}acetamide
3-cyclopentyl-6-[(2,4-dimethoxyphenyl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-[(3-methoxyphenyl)methyl]-8-(oxolane-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-[2-(1H-imidazol-4-yl)ethyl]-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
N-cyclopropyl-5-[(4-ethylpiperazin-1-yl)methyl]-N-propyl-1,2-oxazole-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
2-(4-methoxyphenyl)-5-[(3-methoxypyrrolidin-1-yl)methyl]pyrimidine