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N-[1-(2-methanesulfonylethyl)piperidin-4-yl]-2-methyl-1-benzofuran-5-carboxamide
methyl 2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-6-[3-(methylsulfanyl)propyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{3-cyclopentyl-5-[3-(dimethylamino)propyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
N-(2-ethoxyphenyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
8-methoxy-2-methyl-5-(3-methylpyrazin-2-yl)quinoline
[(3R,4S)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-acetyl-N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}piperidine-3-carboxamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
[(1-ethylpyrrolidin-3-yl)methyl](1H-indol-4-ylmethyl)methylamine
4-{3-[1-(3-methylpyridin-2-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]propyl}morpholine
4-(2,4-dimethoxypyrimidin-5-yl)-N-[2-(dimethylamino)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 4-(4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
4-[2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)ethyl]morpholine
6-(2-chlorophenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
3-(3-chlorobenzoyl)-1-[(3,4-dimethoxyphenyl)methyl]piperidine
4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-2,7,8-trimethylquinoline
5-(2-phenylpyrrolidine-1-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]quinoxaline-5-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N5-methyl-N5-[3-(pyrrolidin-1-yl)propyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-(5-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
2-[2-({methyl[(1-methyl-5-oxopyrrolidin-3-yl)methyl]amino}methyl)phenoxy]acetic acid
5-methanesulfonyl-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
N-{4-[4-(2-methoxy-5-{[methyl(propan-2-yl)amino]methyl}phenoxy)piperidine-1-carbonyl]phenyl}acetamide
(3aR,6aR)-2-acetyl-5-[(3-chloropyridin-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-amine
4-{2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}-3,5-dimethyl-1H-pyrazole
1-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
2-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-butyl-1-(2-methoxyphenyl)-4-(3-methyl-1,2-oxazole-5-carbonyl)piperazin-2-one
2-(3-methylbut-2-en-1-yl)-8-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
N-[2-(piperidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-3-methylthiophene-2-carboxamide
5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-2-(2-methylphenyl)-1,3-oxazole
[3-(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)propyl]dimethylamine
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
3-[(2-hydroxy-3-methoxypropyl)(methyl)carbamoyl]benzoic acid
1-[4-(3-methoxyphenyl)-3-oxopiperazine-1-carbonyl]cyclopropane-1-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]furan-2-carboxamide
2-(4-fluorophenoxymethyl)-4-hydroxy-N-(2-oxopiperidin-3-yl)pyrimidine-5-carboxamide
4-{[(4-ethoxypyrimidin-2-yl)amino]methyl}benzene-1-sulfonamide
2-(dimethyl-1,3-thiazol-5-yl)-1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
1-(5-methyl-1,3-oxazole-4-carbonyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
2-[(4aR,7aS)-4-[3-(3-fluorophenyl)propanoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
N-[(3S,4S)-4-methoxypyrrolidin-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide