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7-{[2-methoxy-5-oxo-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-({1-[2-(9-methyl-9H-carbazol-3-yl)acetyl]piperidin-4-yl}methyl)acetamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propylsulfanyl)ethan-1-one
[(3R,4R)-1-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(1S,4S)-2-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-2-azabicyclo[2.2.1]heptane
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(3-hydroxypropyl)amino]pyridine-3-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-4,5,6,7-tetrahydro-1,3-benzothiazole
(2R)-2-amino-1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methylbutan-1-one
1-(2-hydroxyethyl)-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
6-{[({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]methyl}-1,4-oxazepan-6-ol
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1,8-naphthyridine-2-carboxamide
1-{[1-(hydroxymethyl)cyclobutyl]methyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
1-(5-methanesulfonamido-2-methylphenyl)-3-methyl-3-[(2-methyl-1,3-thiazol-4-yl)methyl]urea
N-[2-(3-fluorophenyl)ethyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-(cyclohexylamino)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-oxo-1-(2-phenylethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
methyl 5-{[(4-fluorophenyl)methyl]amino}-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
1-[cyclohexyl(methyl)amino]-3-[3-({[(4,6-dimethylpyrimidin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
3-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
3-(4-methylpiperazine-1-carbonyl)-N-[(1r,4r)-4-hydroxycyclohexyl]benzene-1-sulfonamide
2-methoxy-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
5-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
8-fluoro-2-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
(2E)-3-(3,4-dimethoxyphenyl)-1-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
1-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methylpiperazine
ethyl 3-({2-[(3-methoxyphenyl)methyl]morpholine-4-carbonyl}amino)propanoate
N-(4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}phenyl)butanamide
(2R,3S,6R)-3-phenyl-5-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
6-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 6-[(oxolan-3-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
6-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-2-carbonitrile
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-2-yl)pyrimidin-4-ol
methyl 3-[(3S,4R)-1-[(2-hydroxy-5-methoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
4-{[3-(methylsulfanyl)phenyl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
2-{[(1R,2S)-2-(methoxymethyl)cyclopentyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(3-methoxypropyl)piperidine
(2S,4R)-N-cycloheptyl-1-{[4-(propan-2-yl)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(2,3-dihydro-1-benzofuran-2-ylmethyl)methylamine
2-methyl-5-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}pyridine
2-(2-chloro-4-fluorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
2-(ethoxymethyl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-(3-hydroxy-4-methylbenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
2-methyl-4-{3-[4-(oxolane-2-carbonyl)-1,4-diazepane-1-carbonyl]phenyl}butan-2-ol
3-(3-methoxypropyl)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidine-3-carboxylic acid
2-{3-[benzyl(methyl)amino]piperidin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide