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7-(1-benzothiophen-3-yl)-4-cyclobutanecarbonyl-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{2-[2-(2-methylphenyl)-1H-imidazol-1-yl]ethyl}-4,5,6,7-tetrahydro-1H-indazole
N-[3-(2-acetyl-5-fluorophenyl)propyl]methanesulfonamide
4-{3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
(1S,4S)-2-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
1-cyclopentyl-4-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperazin-2-one
5-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-(1,4-dioxan-2-ylmethyl)-4-methoxy-N-methyl-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-(4-chlorophenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(3-hydroxypropyl)-9-[2-(2-methylphenoxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[4-(2-methylpropyl)phenyl]methyl}pyrrolidin-3-yl]methanol
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)propanamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-5-phenylpentanamide
9-methoxy-N-methyl-7-oxo-3-[2-(1,3-thiazol-4-yl)acetyl]-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
N-[3-(2-fluorophenyl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-hydroxy-N,N-bis(2-methoxyethyl)-2-methylpyrimidine-5-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)({[2-(methoxymethyl)pyrimidin-5-yl]methyl})(pyridin-3-ylmethyl)amine
6-fluoro-N-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
4-[2-(1H-imidazol-1-yl)ethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-ethoxy-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-methyl-N-{1-oxaspiro[4.4]nonan-3-yl}-4-oxo-4H-3,1-benzoxazine-7-carboxamide
4-hydroxy-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-ethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-pyrazole-4-carboxamide
4-(4-ethoxy-3-methylphenyl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]butan-1-one
[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl](methyl)[(1-methylpyrrolidin-3-yl)methyl]amine
(2S)-2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-3-(4-hydroxyphenyl)propanoic acid
N-(1H-imidazol-2-ylmethyl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
2-[4-(5-ethylthiophene-3-carbonyl)morpholin-3-yl]-1-(thiomorpholin-4-yl)ethan-1-one
7-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-[2-(pyridin-3-ylmethyl)pyrrolidine-1-carbonyl]quinoline
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1,4-diazepane
3-{[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]methyl}-5-methyl-1H-indole-2-carboxylic acid
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
N-(1-methyl-1H-pyrazol-5-yl)-2-[4-propyl-3-(pyridin-3-yl)-1H-pyrazol-1-yl]acetamide
[(5-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-(4-aminoazepan-1-yl)-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
3-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}pyridin-2-amine
5-(2-fluorophenyl)-N-[1-(2-methoxyphenyl)ethyl]-N-methyl-1,2,4-triazin-3-amine
4-[hydroxy(thiophen-2-yl)methyl]-N-(1H-indazol-6-yl)piperidine-1-carboxamide
3-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-ol
N-ethyl-5-(methoxymethyl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-2-carboxamide
4-chloro-1-methyl-N-[(3R,4S)-1-[3-(methylsulfanyl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide