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2-[1-(2H-1,3-benzodioxol-4-ylmethyl)-3-oxopiperazin-2-yl]-N-methylacetamide
3,5-dimethyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1-benzofuran-2-carboxamide
dimethyl[2-(1-{[4-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}piperidin-2-yl)ethyl]amine
1-(2-{1-[3-(difluoromethoxy)benzoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
4-(prop-2-en-1-yl)-N-[4-(propylsulfamoyl)phenyl]piperazine-1-carboxamide
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
6-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
4-benzyl-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
propan-2-yl 4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
9-(6-methylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-benzyl-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
1,3,5-trimethyl-6-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-yl]-3-methanesulfonylpropanamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[5-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
3-[2-oxo-2-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)ethyl]imidazolidine-2,4-dione
ethyl 1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
1-[(2S,3S)-2-amino-3-methylpentanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
2-{[(2-fluorophenyl)methyl](methyl)amino}-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-hydroxyethyl)piperidine-3,5-dicarboxamide
(cyclohex-3-en-1-ylmethyl)(methyl){[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]but-3-en-1-one
7-(cyclopropylmethyl)-2-(2-methyl-1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-fluorophenyl)-1-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propan-1-one
2-({4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methylpyridine
1-[3-chloro-2-(propan-2-yloxy)phenyl]-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)urea
2-(5-{1-[2-(pyridin-3-yloxy)acetyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
4-[1-(4-chlorophenyl)cyclopropanecarbonyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(2-chlorophenyl)methyl]-7-fluoro-N-(2-methoxyethyl)-3-methyl-1H-indole-2-carboxamide
3-[5-(1-phenylcyclopentanecarbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]acetic acid
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
N-(1,4-dioxan-2-ylmethyl)-N,1,3-trimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2-methoxy-4-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)acetamide
2-(furan-2-yl)-1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]azepane
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-2-yl)ethan-1-one
4-chloro-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1H-pyrrole-2-carboxamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[(5-methylfuran-2-yl)methyl]urea
N-[2-(4-methoxyphenyl)phenyl]-1-(1-methylcyclopropanecarbonyl)pyrrolidine-2-carboxamide
(3R,4R)-4-methyl-3-(propan-2-yl)-1-[1-(thiophene-2-carbonyl)piperidin-4-yl]pyrrolidin-3-ol
4-(3-fluoropropyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
2-(2-aminoethyl)-N-(3-chloro-4-phenoxyphenyl)morpholine-4-carboxamide
3-methyl-3-[3-(oxolan-2-yl)propyl]-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
N-{2-[methyl(phenyl)amino]propyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
(4aS,8aR)-6-(1-benzofuran-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-benzyl-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one