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methyl 2-[4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-methyl-2-oxopiperazin-1-yl]acetate
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-(4-{7-methylthieno[3,2-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)acetamide
4,4-difluoro-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-cyclopentyl-9-[2-(4-fluorophenoxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-(1H-1,3-benzodiazole-5-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
2-(cyclohex-1-en-1-yl)-N-{[2-(diethylamino)pyridin-3-yl]methyl}acetamide
2-{1-methyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(4-fluoro-2-methylphenyl)-2-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}acetamide
2-(methylamino)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]acetamide
8-(2-fluorobenzoyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
7-fluoro-3-methyl-N-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1-benzofuran-2-carboxamide
5-[2-(pyridin-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
2-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
3-cyclopropyl-5-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazole
N2-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pyrrolidine-1,2-dicarboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{[3-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N-dimethyl-5-{[8-(6-methylpyridazin-3-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}-1,3-thiazol-2-amine
1-ethyl-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(2R,3R,6R)-5-(2,5-difluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}morpholine
2-[methyl({4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]phenyl})amino]ethan-1-ol
(4aS,7aR)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(2S)-2-aminobutanoyl]-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
1-(3-{[5-methyl-6-(3-phenylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
(2R)-1-{2-methyl-3-[(pyridin-3-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxamide
6-(2-aminoethyl)-N-ethyl-2-methyl-N-(oxolan-2-ylmethyl)pyrimidin-4-amine
2-{2-[4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
N-{[7-(cyclohex-3-ene-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
2-{3-[2-(benzyloxy)ethyl]phenoxy}propanamide
(1s,4s)-N-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
2-(1H-imidazol-2-yl)-N-[1-(methoxymethyl)cyclopentyl]benzamide
1-[(3-methylphenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}acetamide
6,7-dimethoxy-1-[(4-methylphenyl)methyl]-3-[({spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}amino)methyl]-1,2-dihydroquinolin-2-one
3-methyl-7-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
9-[2-(morpholin-3-yl)acetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(5-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
1-{2-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
1-{2-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(5-acetylthiophen-3-yl)-1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethan-1-one
(benzylsulfamoyl)({2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl})amine
5-({2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(2,3-dimethylphenoxy)acetamide
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-[(2-methylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
4-[(2,3-dimethoxyphenyl)methyl]-1,2-dimethylpiperazine
2-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]-2-(2-methoxy-5-methylphenyl)acetic acid