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3-(1H-imidazol-1-ylmethyl)-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine
3-[({1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}oxy)methyl]pyridine
8-[3-(2-methyl-1H-indol-1-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-(2-{1-[5-(hydroxymethyl)furan-2-carbonyl]piperidin-2-yl}ethyl)phenol
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-3-[(4-fluorophenyl)formamido]propanamide
8-[(2-chloro-4-hydroxy-5-methoxyphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{3-[4-(2-oxopyrrolidin-1-yl)piperidine-1-carbonyl]phenoxy}acetamide
1-(methoxymethyl)-N-[(3R,4S)-4-(propan-2-yl)-1-(1H-1,2,3-triazol-4-ylmethyl)pyrrolidin-3-yl]cyclobutane-1-carboxamide
N1-(5-methylpyridin-2-yl)-N3-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}propane-1,3-diamine
N-(3,5-dimethoxyphenyl)-3-[1-(isoquinolin-5-ylmethyl)piperidin-3-yl]propanamide
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperazine
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-{1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-5-phenyl-1H-pyrazole
2-{7-[(2,3-dimethoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxamide
2-chloro-5-acetamido-N-(3-hydroxy-3-phenylpropyl)-N-methylbenzamide
1-[2-(dimethylamino)ethyl]-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
(4aR,7aS)-1-(furan-2-carbonyl)-4-[(2E)-2-methylpent-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{5-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-[(1S,5R)-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-(3,4-dimethoxyphenyl)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(4-methylpiperazin-1-yl)-2-(3-phenoxypropyl)-2,3-dihydropyridazin-3-one
5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-[4-(quinolin-8-ylmethyl)piperazin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-[3-(4-methylbenzenesulfonamido)propyl]-2,3-dihydro-1H-indene-1-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
3-methyl-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridazine
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(2-methoxyphenyl)-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyridazin-3-amine
2-(dimethylamino)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(4-methylphenyl)acetamide
2-(4-acetylphenoxy)-1-[4-(3-fluorophenoxy)piperidin-1-yl]ethan-1-one
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
1-{1-[3-(oxan-4-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
N-[3-(1,3-benzothiazol-2-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[(4-fluorophenyl)methyl]-2-(furan-2-yl)-2-oxo-N-(oxolan-2-ylmethyl)acetamide
4-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}benzonitrile
methyl 9-(cyclopentyloxy)-3-(2-methoxy-2-phenylacetyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(piperidin-1-ylmethyl)cyclopropyl]-1,2-oxazole-3-carboxamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-3,4-dimethoxybenzamide
2-phenyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]imidazo[1,2-a]pyridine-6-carboxamide
6,7-dimethoxy-2-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
2-(2-chlorophenyl)-3-methyl-N-[2-(pyrazin-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
methyl (2R,4S)-4-hydroxy-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine-2-carboxylate
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamide
N-[3-(cyclopentyloxy)phenyl]-4-(pyridin-4-yl)piperazine-1-carboxamide
2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-N-[2-(4-sulfamoylphenyl)ethyl]-1,4-dihydropyridine-3-carboxamide
6-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}piperazin-2-one
4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1λ6-thiomorpholine-1,1-dione
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-9H-purin-6-amine