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N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
3-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
2-{2-[2-(3-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-chlorophenoxy)ethan-1-one
ethyl 1-(1,2-oxazol-3-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-[1-(4-chlorophenyl)cyclobutanecarbonyl]-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aS,6aR)-5-(5-chloropyridin-2-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1R,5R)-6-methyl-3-(2,4,6-trimethylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(6-aminopyridine-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(oxan-4-ylmethyl)acetamide
N-[(3S,4R)-1-(1,3-benzothiazol-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(4aS,7aR)-1-(5-methylthiophene-2-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
3-ethyl-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-ol
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-propylacetamide
N,N-diethyl-1-(5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine
1-(2,6-dimethylpyridin-3-yl)-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
[5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)furan-2-yl]methanol
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-[(3R,4R)-3-hydroxy-1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl]pyrazine-2-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
4-[(3S,5R)-5-[4-(pyridin-4-yl)piperazine-1-carbonyl]piperidine-3-carbonyl]morpholine
6-(2-acetylphenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(pyrrolidin-1-yl)propan-1-one
8-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
[4-({1-[6-(methoxymethyl)pyridine-2-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
4-{[4-(morpholine-4-sulfonyl)phenyl]methyl}-2-(trifluoromethyl)morpholine
2-{[(4-fluoro-3-methylphenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
6-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-3-propyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-{4-[4-(methylamino)pyrimidin-2-yl]phenyl}propanoic acid
N6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]acetamide
N-{[2-(azepan-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)cyclopropanecarboxamide
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
1-(carbamoylmethyl)-N-{[3-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(quinoline-3-carbonyl)pyrrolidin-3-amine
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[3-(3-methoxyphenoxy)azetidin-1-yl]ethan-1-one
ethyl 1-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidine-4-carboxylate
2-({2-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]methyl}-N-methylbenzene-1-sulfonamide
9-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}-N,N-dimethylethane-1-sulfonamide
2-amino-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}ethan-1-one
5-{[1-(cyclohex-1-en-1-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid