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N-tert-butyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-5-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}benzene-1-sulfonamide
7-methyl-3-{[4-(5-propylpyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole
4-(1H-imidazol-2-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine
4-(4-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
N4-[3-(dimethylamino)-1-phenylpropyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-{2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}-1,3-thiazole-4-carboxamide
2-butyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,3-benzoxazole-5-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(oxan-4-yl)piperidine
4,6-dimethyl-2-{4-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperazin-1-yl}pyrimidine
(3aS,6aS)-2-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(3-methylthiophen-2-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[3-(trifluoromethyl)phenyl]ethan-1-one
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-(2-aminoethyl)-N,5,6-trimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
N-(2-hydroxyethyl)-3-[5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
2-(7-chloro-4-hydroxyquinoline-3-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[2-(2-methoxy-4-methylphenoxy)ethyl]-4-(pyrrolidin-1-yl)piperidine
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-ethoxy-1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
3-({[(3-fluorophenyl)methyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
3-methyl-6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridazine
1-methyl-5-{[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]sulfanyl}-1H-1,2,3,4-tetrazole
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-{1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidin-4-yl}-1,4-diazepan-5-one
6-(2-methoxybutyl)-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-methyl-1-[(2-methylphenyl)methyl]-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-({5-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]-2-methoxyphenyl}methyl)-1H-1,2,4-triazole
3-{6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-3,9-diazaspiro[5.6]dodecan-10-one
2-chloro-N-({1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-3-yl}methyl)benzamide
(1S,5R)-6-benzyl-3-[2-(4-fluorophenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-methoxypropyl)-6-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-(1-methyl-1H-pyrazol-5-yl)-2-{3-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}acetamide
6-[({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-3-carbonitrile
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
1-(2-methoxy-5-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
(3R,4S)-1-[2-(2-methoxy-4-methylphenoxy)ethyl]-3,4-dimethylpiperidin-4-ol
3,6-dimethyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1-benzofuran-2-carboxamide
1-(5-ethylthiophene-3-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(phenylsulfanyl)ethan-1-one
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
(1S,5R)-6-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
butyl 1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxylate
5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-cyclobutanecarbonyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]piperidine-4-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}pyrrolidine-3-carboxylic acid
N-[2-(2,4-dimethylphenoxy)ethyl]-N-methyl-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide