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1-[1-(3-aminopropanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(3S)-N,N-dimethyl-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)azepan-3-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2,5-dimethylfuran-3-carboxamide
3-(2-chlorophenoxy)-1-(oxolan-3-ylmethyl)azetidine
3-(3-fluorophenoxymethyl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]propanamide
2-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
3-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine
4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}piperidin-2-one
2-methyl-4-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)-6-(pyrrolidin-1-yl)pyrimidine
3-[4-(azocan-1-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl]-1H-indole
2-{4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperazin-1-yl}pyrazine
[(2-chlorophenyl)methyl][(8-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}quinolin-3-yl)methyl]amine
ethyl 5-{[2-methoxy-2-(thiophen-2-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylate
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-1,3-thiazole-5-carboxamide
1-{5-[1-(piperidin-1-yl)ethyl]furan-2-carbonyl}-4-(pyridin-4-yl)piperazine
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(3,4-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
methyl 2-[(2-methoxyethyl)(thiophen-2-ylmethyl)carbamoyl]benzoate
N-(2-hydroxyethyl)-3-[5-(2-methylfuran-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
4-chloro-2-[3-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]phenol
6-methoxy-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
dimethyl({[4-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-2-yl)phenyl]methyl})amine
2-(3-chloro-2,4-difluorophenyl)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
2-ethoxy-N-[(3R,4S)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-[2-amino-4-methyl-6-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)pyrimidin-5-yl]propanoic acid
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(4-hydroxyphenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-[(4-methylphenyl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-amino-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-4-phenyl-1H-pyrazole-3-carboxamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(furan-2-ylmethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
8-(butan-2-yl)-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclohexyl-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-[4-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)morpholin-3-yl]acetic acid
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(cyclohexylmethyl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N2,N2-dimethyl-N4-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-(4-methanesulfonylphenyl)-5-propylpyrimidine
4-[2-(furan-2-yl)-1H-imidazol-1-yl]-1-methanesulfonylpiperidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
{2-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}urea
2-[3-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]ethan-1-ol
1-(2,3-dimethoxyphenyl)-2-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3-methyl-1-(2-methylpropyl)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperazin-2-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
2-methyl-N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)-1,3-thiazole-4-carboxamide
N-{1-[1-(4-chlorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
3-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}phenol