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N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(4-methyl-1,4-diazepan-1-yl)-N-(propan-2-yl)acetamide
(2S)-2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}-3-phenylpropanamide
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
3-(1-ethyl-1H-imidazol-2-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidine
4-(5-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}furan-2-carbonyl)morpholine
2-(naphthalen-2-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2-methylphenyl)benzamide
2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-[(5-methylfuran-2-yl)methyl]acetamide
2-{3-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]piperidin-1-yl}acetamide
1,5-dimethyl-4-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
ethyl 4-(2,3-dihydro-1H-indene-1-amido)piperidine-1-carboxylate
2-(4-fluorophenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-4-hydroxy-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(quinolin-8-yloxy)ethyl]acetamide
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1,3-dimethyl-N-[1-(6-methylpyridin-2-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(dimethyl-1,3-thiazol-5-yl)-1-[2-(3-methoxyphenyl)azetidin-1-yl]ethan-1-one
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(thiophen-2-ylmethyl)amine
N3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
2-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]pyridine-4-carbonitrile
2-methyl-1-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}azetidin-3-yl)piperidine
4-{4-[(4-methoxyphenyl)methyl]-3-oxopiperazine-1-carbonyl}benzonitrile
3-fluoro-2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
(3ar,6ar)-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-methyl-2-(pyridin-4-yl)-N-(quinolin-8-ylmethyl)pyrimidine-5-carboxamide
4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-N-(4-methoxyphenyl)piperidine-1-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclohexyl-3-{[1-(3,5-difluorophenyl)ethyl]amino}propanamide
[(2-chloropyridin-3-yl)methyl][(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]methylamine
6-[(3-chloro-1H-indol-2-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-benzyl{[2-(1H-pyrrol-1-yl)phenyl]amino}sulfonamide
(1R,7S)-3-(4-fluoro-2-methylphenyl)-N-methyl-4-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]acetamide
N-cyclopropyl-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperazine-2-carboxamide
1-{[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(oxolan-3-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-[(3R,4S)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-propylpyrrolidin-3-yl]cyclobutanecarboxamide
1-[3-(difluoromethoxy)benzoyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
3-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
ethyl 1-(2,4-dimethylphenyl)-5-{[(1,2-oxazol-3-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
6-(3-fluoro-4-methoxyphenyl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
1-cyclohexyl-N5-cyclopropyl-N3-[(3-methoxyphenyl)methyl]-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-(4-methyl-2-oxo-2H-chromen-7-yl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-fluoro-N-[4-(4-{[2-hydroxy-3-(3-methoxyphenoxy)propyl]amino}piperidin-1-yl)phenyl]benzamide
N'-ethyl-N'-[2-(piperidin-1-yl)ethyl]-N-(2,4,6-trimethylphenyl)butanediamide
1-benzyl-8-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione