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4-benzyl-3-ethyl-1-(pyrrolidine-1-sulfonyl)-1,4-diazepan-5-one
4-chloro-1,5-dimethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-3-carboxamide
3-butyl-1-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)urea
(3aR,6aR)-2-cyclopentanecarbonyl-5-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(prop-2-en-1-yl)(prop-2-yn-1-yl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
(1s,4s)-4-(3-benzoylpiperidine-1-carbonyl)cyclohexan-1-ol
(2R)-2-amino-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methoxypropanamide
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propyl-5-{1-[2-(thiophen-2-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N-(3-ethoxy-2-hydroxypropyl)-4-{[(4-methylphenyl)amino]methyl}benzamide
N-[2-(oxan-2-yl)ethyl]-6-(propan-2-yl)pyrimidin-4-amine
4-({2-[(benzenesulfonyl)methyl]phenyl}methyl)-1,4-oxazepan-6-ol
4-methoxy-6-[3-(methoxymethyl)pyrrolidin-1-yl]pyrimidin-2-amine
N-{2-[2-(1H-imidazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
6-{3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
N-(furan-3-ylmethyl)-N-methyl-4-(4-methylphenoxy)piperidine-4-carboxamide
1-(oxolan-3-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methylpropanamide
N,N-dimethyl-4-({3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)aniline
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
methyl 3-{[(1-methyl-1H-pyrazol-5-yl)formamido]methyl}-5-[3-(trifluoromethyl)benzamido]benzoate
N-[4-chloro-2-(trifluoromethyl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-(2,4,5-trimethoxybenzoyl)piperidine
(3R,4R)-4-(azepan-1-yl)-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-3-ol
4-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
(3S)-1-(3,5-dimethyladamantane-1-carbonyl)pyrrolidin-3-ol
[3-(2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]dimethylamine
2-methyl-6-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-[(3-fluorophenyl)methyl]morpholine
5-(1H-indol-2-ylmethyl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 2-[2-(4-chlorophenyl)morpholin-4-yl]pyridine-3-carboxylate
8-(2-methyl-5-propylpyrimidin-4-yl)-1-oxa-8-azaspiro[4.5]decane
1-(3,6-dimethylpyrazin-2-yl)-3-(2-phenoxyethyl)piperidine-3-carboxylic acid
3-methyl-8-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
1-(2-aminoethyl)-N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
1-(pyridin-2-ylmethyl)-4-[4-(pyridin-4-yl)piperazine-1-carbonyl]pyrrolidin-2-one
4-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}-N-methylbenzene-1-sulfonamide
3-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]quinoline-4-carboxylic acid
dimethyl[3-(4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)propyl]amine
1-(8-fluoroquinoline-2-carbonyl)-4-(hydroxymethyl)azepan-4-ol
(1S,4S)-2-(3-chlorophenyl)-5-[(5-methylthiophen-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
methyl 1-{2-hydroxy-3-[3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
7-[(2S)-2-(dipropylamino)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-6-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
2-[4-chloro-2-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]acetamide