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4-cyano-N-[(3R,4S)-1-(furan-2-ylmethyl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
5-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-methoxyphenyl)-N-methyl-1,3-benzoxazole-6-carboxamide
2-(dimethylamino)-1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-(3-methylphenyl)ethan-1-one
4-(5-ethyl-2-methylpyrimidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{1-[2-(1,3-benzoxazol-2-yl)acetyl]piperidin-3-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2,5-dichloro-N-{2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}benzamide
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(1H-imidazol-1-ylmethyl)piperidine
N-(1-benzylcyclopropyl)-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-[3-(2-methoxyethyl)-5-(3-methyl-4-oxo-3,4-dihydroquinazolin-7-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(2-methylpyrimidin-4-yl)piperidin-3-amine
7-cyclopentyl-2-(pyridazine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(propan-2-yl)({[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-methyl-N-{2-[methyl(phenyl)amino]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
ethyl 4-(6-methyl-3-{[(thiophen-2-ylmethyl)amino]methyl}quinolin-2-yl)piperazine-1-carboxylate
1-(furan-2-ylmethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]piperidine-3-carboxamide
2-methyl-1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
1-[4-(4-methylphenoxy)piperidin-1-yl]-2-(morpholin-3-yl)ethan-1-one
1-{2-oxo-2-[3-(phenylamino)piperidin-1-yl]ethyl}piperidin-2-one
methyl 3-(dimethyl-1,2-oxazole-4-carbonyl)-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-({5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-1,2-dihydroisoquinolin-1-one
N-{[4-(dimethylamino)oxan-4-yl]methyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-oxo-N-(propan-2-yl)acetamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[3-(8-chloroquinolin-2-yl)phenyl]ethan-1-one
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]propanamide
methyl 3-cyclobutaneamido-5-{[(4-methylphenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[2-(4-fluorophenyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]thiomorpholine
1-ethyl-N-(pyridin-4-ylmethyl)-5-[(thiophen-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(3-fluorophenyl)-1-(3-methoxypiperidin-1-yl)propan-1-one
(3S,9aR)-3-benzyl-8-(2,5-dimethylbenzenesulfonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[4-(4-fluorophenoxy)phenyl]-3-[3-(4-hydroxypiperidin-1-yl)propyl]urea
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
(5S,9aS,9bS)-5-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[3-(azepan-1-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2,1,3-benzothiadiazol-5-ylmethyl)({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-({[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyridine
4-({4-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]furan-2-yl}methyl)morpholine
7-fluoro-3-{[2-(furan-2-yl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(3-hydroxyquinoxalin-2-yl)propanamide
4-hydroxy-4-(hydroxymethyl)-N-(2,3,5-trifluorophenyl)azepane-1-carboxamide
2-butyl-N-(2-chloropyridin-3-yl)-4-methyl-3-oxopiperazine-1-carboxamide
N-[2-(4-fluorophenyl)-1-[1-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]ethyl]-2-methoxy-N-methylacetamide
2-(methylsulfanyl)-3-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]pyridine