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3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-methyl-3,4-dihydroquinazolin-4-one
4-[({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]benzonitrile
9-(5-chloro-2-methoxybenzoyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
5-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-2-(3-methoxyphenyl)piperidine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]pyrrolidin-3-yl]acetamide
5-(3-cyclopropylpropanoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{[1-(5-chloro-2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1H-1,2,3,4-tetrazole
N-methyl-4-[6-(trifluoromethyl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,4R)-1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
6-(2-chlorophenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)[1-(pyridin-3-yl)propyl]amine
(1S,6R)-9-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
2-[(3R,4S)-3-[(2-aminopyrimidin-4-yl)amino]-4-propylpyrrolidin-1-yl]-1-(piperidin-1-yl)ethan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]butanamide
1-(3-chlorophenyl)-4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperazin-2-one
3-(2,5-dihydroxy-2-methylpentyl)-1-(2-fluoro-4-methoxyphenyl)urea
5-[2-(4-fluorophenyl)azetidine-1-carbonyl]-3-(2-methylpropyl)-1,2-oxazole
4-(4-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
3-butyl-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-methylpiperazin-2-one
4-{[1-(3-phenylpropyl)piperidin-3-yl]carbamoyl}pyridin-1-ium-1-olate
N-(diphenylmethyl)-1-ethyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-methyl-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-3-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridin-4-one
5-(methoxymethyl)-N-[1-(thiophen-2-yl)ethyl]furan-2-carboxamide
(2R)-3-hydroxy-2-[4-phenyl-5-(trimethyl-1H-pyrazol-4-yl)-1H-imidazol-1-yl]propanoic acid
7-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
2-[(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
3-methoxy-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
2-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-benzyl-N-methyl-1,2-oxazole-3-carboxamide
N-[(3,5-difluorophenyl)methyl]-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
1-(benzyloxy)-8-[2-(1,3-thiazol-4-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
5-{[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-3-(3-methoxyphenyl)-1,2-oxazole
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]-1,2-dihydropyrimidin-2-one
1-{5-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}quinoline-4-carboxylic acid
N-(3-methoxypropyl)-4-methyl-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
5,7-dimethyl-N-(oxan-4-yl)pyrido[2,3-d]pyrimidin-4-amine
N-[4-(1H-indol-2-yl)phenyl]-4-(2-methoxyethyl)piperazine-1-carboxamide
8-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}sulfonyl)quinoline
3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-1-[(2-chlorophenyl)methyl]-7-methoxy-1,2-dihydroquinolin-2-one
N,N-dimethyl-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)benzoyl]pyrrolidin-3-amine
N-phenyl-5-[2-(1H-1,2,4-triazol-3-ylsulfanyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1'-(2-methyl-5-propylpyrimidin-4-yl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]