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N,1-dimethyl-6-oxo-N-(quinolin-3-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}acetamide
5-{4-hydroxy-1-[(3-methylphenyl)methyl]piperidin-4-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
3-ethyl-4-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]piperazin-2-one
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
1-(cyclopropylmethyl)-5-(2-methoxypyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[(4H-1,2,4-triazol-4-yl)carbamoyl]adamantan-1-yl acetate
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]but-2-ynamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-methyl-1H-1,3-benzodiazole-4-carboxamide
methyl 4-{[1-methyl-2,4-dioxo-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
2-(5-fluoro-2-methylphenyl)-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetic acid
4-ethyl-3-(piperidin-4-yl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-methyl-6-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}ethan-1-amine
(1S,5R)-3-(quinoxalin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-fluorophenyl)-2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]acetic acid
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroquinolin-2-one
1-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
1-[7-(3-chlorophenyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
5,6-dimethoxy-2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,2-dihydroisoquinolin-1-one
N-(furan-3-ylmethyl)-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
(2R,3R)-2-amino-1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-methylpentan-1-one
2-{[(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amino]methyl}benzoic acid
6-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carbonitrile
2-methyl-4-(4-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}phenyl)butan-2-ol
4-[(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]morpholine
5-{2-[2-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)amino]methyl}piperidin-2-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
2-ethyl-5-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,3,4-oxadiazole
N3-benzyl-N5-(1-benzylpyrrolidin-3-yl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-[3-(4-methyl-1,3-thiazol-5-yl)-1H-pyrazol-1-yl]acetamide
2,2-dimethylpropyl (2S,4S)-4-fluoro-2-(methanesulfonamidomethyl)pyrrolidine-1-carboxylate
4-hydroxy-2-methyl-N-{1-oxaspiro[4.5]decan-3-yl}pyrimidine-5-carboxamide
(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(methoxymethyl)-6-[3-(2-methylpropoxy)phenyl]pyrimidine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
2-(4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
2-butyl-8-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(3,4-dimethoxyphenyl)methyl]-N-[(3-methyloxetan-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-[2-(3-methylpyridin-2-yl)ethyl]-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
2-ethyl-9-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(2,3,4-trimethoxyphenyl)quinoline
(1R)-2-(1H-indol-3-yl)-1-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethan-1-amine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(oxolan-3-ylmethyl)sulfamoyl]benzamide
2-(3-chlorophenoxy)-N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-{4-[4-(methoxycarbonyl)phenyl]piperazin-1-yl}pyridine-4-carboxylic acid
2-propyl-N-[2-(1H-pyrrol-1-yl)ethyl]-1,3-thiazole-4-carboxamide
3,3-dimethyl-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]but-2-yn-1-one