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6-(3-fluorophenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
(4aS,8aR)-1-butyl-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
(2S)-N-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
2-(4-hydroxyphenyl)-2-[4-(3-methoxybenzoyl)piperazin-1-yl]acetic acid
3-({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)-N-(1,3-thiazol-2-yl)propanamide
N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-4-carboxamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
3-(aminomethyl)-N-{3-chloro-4-[(propan-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide
2-methoxy-3-{[(oxolan-3-yl)amino]methyl}-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3,3-dimethyl-1-[(3S,4R)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
5-{1-[(3S,4R)-4-methoxyoxolan-3-yl]-4-phenyl-1H-imidazol-5-yl}-3-phenyl-1,2,4-oxadiazole
1-(5-{6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}-1H-1,2,4-triazol-1-yl)butan-2-ol
2-[1-(4-methanesulfonylbenzenesulfonyl)azetidin-3-yl]pyridine
N-(furan-2-ylmethyl)-8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2,4-dimethyl-N-{4-[4-(thiomorpholin-4-yl)piperidin-1-yl]phenyl}benzamide
1-methyl-N-{3-[methyl(phenyl)amino]propyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1-ethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-benzyl-4-(2-methylpyridine-3-carbonyl)morpholine
N-(2,2-difluoroethyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}benzamide
2-[N-(4-methylphenyl)methanesulfonamido]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]acetamide
2-[3-cyclopropyl-5-(3-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
N-cyclopentyl-2,2-dimethyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)oxane-4-carboxamide
N-[3-({[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
7-fluoro-3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
2-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
7,7-dimethyl-2-[1-(pyridin-2-yl)piperidin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-acetyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)thiophene-2-carboxamide
(3S,4S)-1-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-(oxolan-2-ylmethyl)-1-(thiophen-3-ylmethyl)urea
3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
2-[(cyclopropylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
[(5-{[(1-ethyl-1H-indol-3-yl)sulfanyl]methyl}-1,2,4-oxadiazol-3-yl)methyl]dimethylamine
(1R,2R,6S,7S)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-(2-ethyl-1H-1,3-benzodiazol-6-yl)-1-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
(3R,4R)-3-cyclopropyl-1-(4-ethyl-5-methylpyrimidin-2-yl)-4-methylpyrrolidin-3-ol
N-[3-(3-fluorophenyl)phenyl]-1-[(3-hydroxyphenyl)methyl]piperidine-4-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
2,3-dimethyl-6-[3-(pyridin-2-yl)azetidine-1-carbonyl]quinoxaline
1-(cyclohexylmethyl)-3-hydroxy-3-{[(prop-2-en-1-yl)amino]methyl}piperidin-2-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4R)-4-amino-N-methyl-1-[2-(phenylamino)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
2-[(4-chlorophenyl)methyl]-5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(3-chloro-4-fluorophenyl)-1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
3-[(3R,4S)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-methanesulfonyl-N,2-dimethylpyrimidin-4-amine