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1-ethyl-8-[(2-methoxyquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R)-5-oxo-N-{2-[(pyridin-2-ylmethyl)carbamoyl]phenyl}pyrrolidine-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(2-phenylethyl)benzamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)quinoline-2-carboxamide
(1R,2R,6S,7S)-4-(trimethylpyrimidin-4-yl)-4-azatricyclo[5.2.1.02,6]decane
3-{5-[1-(2-methoxyacetyl)-4-methylpiperazine-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
3,5-dimethyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1,2-oxazole-4-sulfonamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridine-2-carbonitrile
1-(3-methoxypropyl)-8-{[4-(methylsulfanyl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(5-fluoro-3-methyl-1H-indol-2-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-5-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
(2S,4S)-4-amino-N-methyl-1-[2-(phenylamino)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-(propan-2-yl)piperidine-1-carboxamide
3-{2-[(dimethylamino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-8-fluoro-1,4-dihydroquinolin-4-one
4-(2,3-dihydro-1,4-benzodioxin-6-yl)thiophene-2-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
(3S)-1-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrrolidin-3-ol
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(3-phenylpropyl)acetamide
2-methyl-4-propyl-6-{4-[4-(pyridin-4-yl)piperazin-1-yl]piperidin-1-yl}pyrimidine
2-(4-fluorophenyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
(3aR,7aS)-5-methyl-2-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-(6-methylpyridazin-3-yl)benzoic acid
methyl 3-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}benzoate
4-methyl-6-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidin-2-amine
4-(1H-imidazol-1-ylmethyl)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-ol
4-{2-[1-(2,5-difluorobenzenesulfonyl)piperidin-2-yl]ethyl}morpholine
4-cyclobutyl-6-methyl-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrimidine
1-{2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
7-(2-ethoxyethoxy)-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1,2,3,4-tetrahydroquinolin-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-2-methylfuran-3-carboxamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyridin-2-amine
14-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
5-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-2-amine
4-{[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
2-ethyl-9-[(3-methylquinoxalin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2,6-dimethoxy-N-methylpyridine-3-carboxamide
3-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)pyridin-2-amine
1-{3-[3-(benzyloxy)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
3-({2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[5-(methoxymethyl)furan-2-carbonyl]-3-(naphthalene-2-carbonyl)piperidine
(2R)-2-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)pyrrolidine-2-carboxamide
4-{ethyl[4-(4-fluorophenyl)butyl]amino}butan-1-ol
1-[(5-methylpyrazin-2-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
N-[3-(4-methoxyphenyl)propyl]-6-(3-methoxypiperidin-1-yl)pyridine-3-carboxamide
N-(1-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide