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N-benzyl-N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
N,2-dimethyl-5-phenyl-N-(pyrazin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-[3-(furan-2-yl)propanoyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
7-(2-cyclohexylethyl)-2-[2-(1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-[2-methoxy-4-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
(1S,2S)-2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclohexan-1-ol
7-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)thiophene-2-carboxamide
3-(2-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-2-(4-oxo-1,4-dihydroquinolin-1-yl)acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidine-3-carboxylic acid
N-cyclopentyl-3-{[(1H-indazol-7-yl)carbamoyl]methyl}morpholine-4-carboxamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-oxo-2H-pyran-5-carboxamide
1-(4-{2-methoxy-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-N-methylmorpholine-2-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
6-{[5-(2-chlorophenyl)furan-2-yl]methyl}-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(ethylamino)-N-[2-(3-phenylpiperidin-1-yl)ethyl]pyrimidine-5-carboxamide
N-cyclopentyl-4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)benzamide
(3E)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]pent-3-en-1-one
(1R,3S)-7-[2-(2,4-dimethylphenoxy)ethyl]-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
N-(pyridin-2-ylmethyl)-4-({1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
1-{3-[(4-cyclohexylpiperazin-1-yl)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
2-(hydroxymethyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
(2R,3R)-3-amino-1'-(4-hydroxybenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-{3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]phenyl}-1H-1,2,3,4-tetrazole
(3aR,6aR)-2-cyclopentyl-5-[(4,6-dimethylpyrimidin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)urea
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
4-benzyl-3-(piperidin-4-yl)-1-(quinolin-8-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
2-ethyl-6-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidin-4-amine
2-methyl-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(pyrrolidin-1-yl)propan-1-one
1-{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}-3-(2-methylphenyl)pyrrolidin-3-ol
1-[(2-fluorophenyl)methyl]-4-[1-(hydroxymethyl)cyclopropanecarbonyl]-1,4-diazepan-6-ol
(3R,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-(3-phenylpropyl)pyrrolidin-3-amine
(2R,3R)-3-{[2-(2-ethylphenoxy)ethyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[2-(morpholin-4-yl)ethyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-1-carboxamide
4-(naphthalen-2-ylmethyl)-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
2-(methylsulfanyl)-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-cyclohexyl-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-4-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-(2-phenyl-1H-imidazol-1-yl)-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}ethan-1-one
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-[1-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)piperidin-3-yl]propan-1-ol
9-(cyclopropylmethyl)-4-(2,4-dimethylpyrimidine-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one