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1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methoxy-2-methylpropan-1-one
(1S,2S)-2-{4-[(6-methylpyridin-3-yl)methyl]piperazin-1-yl}cyclohexan-1-ol
2-methyl-3-[(pyridin-2-ylmethyl)amino]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
9-ethyl-1-methyl-4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-[3-(morpholin-4-yl)azetidin-1-yl]butan-1-one
N-[4-fluoro-3-(methylcarbamoyl)phenyl]-4-(3-methoxyphenyl)piperazine-1-carboxamide
3-butyl-1-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-{3-[(2,6-dichlorophenyl)methyl]-1-ethyl-1H-1,2,4-triazol-5-yl}-1λ6-thiolane-1,1-dione
7-{3-[5-(4-methylphenyl)furan-2-yl]propanoyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-[(1S,5S)-3,6-diazabicyclo[3.2.2]nonan-3-ylmethyl]-1H-1,3-benzodiazole
N-methyl-N'-(4-methylphenyl)-N-(quinolin-3-ylmethyl)propanediamide
3-[(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
5-{2-[(5-methylhex-5-en-2-yl)amino]ethyl}-1,3,4-thiadiazol-2-amine
6-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-N-propylpyridine-3-carboxamide
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
1-{2-[4-(1,2-oxazolidine-2-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperidine
1-[(5-methoxy-1H-indol-2-yl)methyl]-3-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]urea
8-(3-hydroxypropyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-cyclopropylpropan-1-one
N-methyl-4-(4-methylphenyl)-N-[(3-methylpyridin-4-yl)methyl]-5-(pyridin-4-yl)pyrimidin-2-amine
N-(butan-2-yl)-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
2-({[2-(2-methylphenoxy)pyridin-3-yl]methyl}amino)pyridine-4-carbonitrile
3-amino-1-(4-cyclohexyl-1,4-diazepan-1-yl)-3-phenylpropan-1-one
1-[4-(4-methylphenoxy)piperidin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-(2-hydroxy-3-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-3-(3,6-dimethyl-1-benzofuran-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-(4-methoxyphenyl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-methoxyethyl)-4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazine
7-[(3-methyl-1-benzofuran-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-(3-chloro-4-fluorophenyl)-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}propanamide
(3aS,7aR)-5-methyl-2-(1-methyl-1H-indole-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-{4-[(3-methoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(2-methylphenyl)methyl]pyrrolidin-2-one
4-[5-(2-methyl-1-benzofuran-7-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]morpholine
4-(pyrrolidin-1-ylmethyl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
8-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-methylfuran-2-yl)methyl]-3-[1-(1H-pyrazole-4-sulfonyl)piperidin-3-yl]propanamide
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
3-(2,5-dimethyl-1H-pyrrol-1-yl)-4,5-dimethyl-N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]thiophene-2-carboxamide
N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
1-{5-[(2-amino-6-methylpyrimidin-4-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
3-cyclopentyl-1-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(thiophen-3-ylmethyl)urea
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-4-(piperidin-1-ylmethyl)benzamide
4-({4-[3-(3,3-diethylpyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
2-{4-[4-(cyclopropylcarbamoyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-4-carboxamide
3-[(dimethylamino)methyl]-N-[1-(methoxymethyl)cyclopentyl]benzamide
2-(4-methyl-6-{[3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-2-yl)phenol