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3-({1-[(4-fluoro-3-methylphenyl)methyl]piperidin-4-yl}oxy)pyridine
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-[(2-methylpyrrolidin-1-yl)sulfonyl]benzamide
ethyl 1-{[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]carbamoyl}-4-oxopiperidine-3-carboxylate
N-(4-fluoro-2-methylphenyl)-3-{1-[3-(2-fluorophenyl)propanoyl]piperidin-3-yl}propanamide
7-methyl-N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
ethyl 4-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-amido}piperidine-1-carboxylate
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(6-phenoxypyridin-3-yl)piperidine-1-carboxamide
3-[2-(dimethylsulfamoyl)ethyl]-1-[3-methoxy-5-(trifluoromethyl)phenyl]urea
2-ethoxy-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
1-ethyl-3-(2-methylpropyl)-N-(2-oxopyrrolidin-3-yl)-1H-pyrazole-5-carboxamide
3-({1-[(2-methylpyrimidin-5-yl)methyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)propanamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]pyrrolidin-3-yl]methanol
2-{2-[(3,3-dimethylpyrrolidin-1-yl)methyl]phenyl}-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
6-cyclopentyl-N-[2-(ethanesulfonyl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(thiophen-2-ylmethyl)acetamide
N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
8-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
5-(2-cyclopropyl-1,3-benzoxazole-6-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[2-(pyridin-4-yl)ethyl]propanamide
2-(dimethylamino)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
2-amino-4-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}quinazoline-6-carboxylic acid
N-[1-(1-cyclohexylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxybenzamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]acetamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
5-methyl-N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
5-(4-methyl-1,4-diazepan-1-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-methyl-3-(2-oxopyrrolidin-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
2-{4-methyl-6-[(oxolan-3-yl)amino]pyrimidin-2-yl}phenol
N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 4-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}thiophene-2-carboxylate
3-[5-(1-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-1H-imidazol-2-yl)thiophen-3-yl]prop-2-yn-1-ol
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]piperidin-1-yl}-5-ethyl-2-methylpyrimidine
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-8-fluoroquinoline-2-carboxamide
1-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
ethyl({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-3-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-propoxyacetamide
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
1-(3-fluorobenzenesulfonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
7-{[4-(propan-2-yl)phenyl]methyl}-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2,4-dimethyl-7-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
1-[3-({[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]ethan-1-one
3-fluoro-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-[3-(methylamino)propyl]-4-{[2-(1H-pyrazol-4-yl)ethyl]sulfamoyl}benzamide