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1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]piperazine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(6-methylpyridazin-3-yl)pyrrolidin-3-yl]acetamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]but-3-enamide
methyl 3-({1-[(2-methoxyphenyl)methyl]-5-[(3-methylbutyl)carbamoyl]-4-oxo-1,4-dihydropyridin-3-yl}formamido)propanoate
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(6-hydroxypyrimidin-4-yl)methyl]propanamide
N-(1H-indol-4-ylmethyl)-3-(1,2-oxazinan-2-yl)propanamide
(2E)-3-(2-chlorophenyl)-N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(pyridin-4-ylmethyl)prop-2-enamide
6-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]hexan-1-ol
2-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-6-methylphenol
2-[4-(4-{[3-(1H-imidazol-1-yl)-1-phenylpropyl]amino}piperidin-1-yl)phenyl]-1-(pyrrolidin-1-yl)ethan-1-one
2-(4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrazine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}-2-(3-phenylpropyl)morpholine
[(3R,5R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
1-[1'-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2-methyl-1,4-diazepan-5-one
2-(4-ethylpiperazin-1-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
N-[(5-chloro-1H-indol-2-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(butan-2-yl)[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl](pyridin-3-ylmethyl)amine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[2-(1H-imidazol-4-yl)ethyl]propanamide
4-[5-(1-cyclopentanecarbonylpyrrolidin-2-yl)thiophene-2-carbonyl]-1,4-oxazepane
2-[N-cycloheptyl-1-(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]acetic acid
1-{6-azaspiro[2.5]octane-1-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(4aR,8aS)-1-[2-(1H-pyrazol-1-yl)benzoyl]-6-(thiophene-2-carbonyl)-decahydro-1,6-naphthyridine
1'-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-cyclopentyl-N-cyclopropyl-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}acetamide
2-benzyl-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,3-thiazole-4-carboxamide
methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})[1-(pyridin-3-yl)ethyl]amine
(3R,4R)-3-cyclopropyl-1-[(3,5-dichloropyridin-4-yl)methyl]-4-methylpyrrolidin-3-ol
1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
2-(3-{[4-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
1-[7-(2-methoxyacetyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine-3-carboxamide
2-(4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)-1,3-benzoxazole
N-benzyl-N-(cyclobutylmethyl)-2,6-dimethylpyridine-4-carboxamide
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-[(2-phenylethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-{2-[(dimethylamino)methyl]phenyl}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
4-(furan-2-ylmethyl)-3-(pyrazin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-benzyl-N3-[(1-hydroxycyclohexyl)methyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-chloro-N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
1-(3,5-dimethylphenyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-2-one
4-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
N,1-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
3-[3-(furan-2-yl)propyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
6-(propan-2-yl)-N4-[2-(1,3-thiazol-4-yl)ethyl]pyrimidine-2,4-diamine
methyl (1R,5S,6R)-6-{[4-(2-ethylphenyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
1-[2-(3,4-dimethylphenyl)pyrimidin-4-yl]pyrrolidin-3-ol
4-{[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}-N-(furan-2-ylmethyl)pyridine-2-carboxamide
2-tert-butyl-1,3-dioxo-N-[2-(pyrazin-2-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
5-(2,4-dimethoxybenzoyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine