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5-[3-cyclopropyl-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-2-(methylsulfanyl)pyrimidine
3-(cyclopropylmethyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxylic acid
(1S,5R)-6-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(2,3-difluorophenyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[2-(2-ethoxyphenyl)ethyl]-8-fluoroquinoline-2-carboxamide
benzyl({[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl})ethylamine
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
3-{1-[(2-ethylphenyl)methyl]piperidin-3-yl}propanamide
4-{[1-(2,3-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiane-1,1-dione
N-methyl-N-(3-phenylpropyl)-5-propyl-1,3,4-oxadiazole-2-carboxamide
[4-(4-{1-[(2-methoxypyrimidin-5-yl)methyl]pyrrolidin-3-yl}pyridin-2-yl)phenyl]methanol
[(3-methoxyphenyl)methyl](prop-2-en-1-yl){[1-(propan-2-yl)piperidin-4-yl]methyl}amine
N-(1-{4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}cyclopentyl)aniline
2-(3,4-dichlorophenyl)-4-(5-ethyl-2-methylpyrimidin-4-yl)morpholine
2-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
4-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
2-[2-(2,2-diphenylethyl)morpholin-4-yl]acetic acid
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-(1H-pyrazol-3-yl)benzamide
8-benzyl-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N3-(1-benzothiophen-2-ylmethyl)-1-(cyclohexylmethyl)-N3,N5,N5-trimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-(1-benzofuran-5-yl)-1-[(3S,4R)-4-methoxyoxolan-3-yl]-4-phenyl-1H-imidazole
4-(1-methyl-1H-imidazol-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine
3-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-4-[(3-methylphenyl)methyl]piperazine
butyl 4-(furan-2-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
5-{[5-(oxan-2-yl)furan-2-yl]methyl}-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3,5,7-trimethyl-N-[3-(3-oxopiperazin-1-yl)propyl]-1H-indole-2-carboxamide
1-[3-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-(3-methyl-1H-pyrazol-1-yl)-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
1-[(3S,4R)-1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
6-(4-fluorophenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[2-(2-fluorophenyl)ethyl]piperidine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}cyclohexanecarboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(4,6-dimethyl-2-oxo-2H-pyran-5-carbonyl)-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
N-[2-(dimethylamino)ethyl]-3-[1-(5-hydroxypyridine-2-carbonyl)piperidin-4-yl]propanamide
N-cyclohexyl-N-methyl-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)azepane
N-(3,4-dimethylphenyl)-1-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)piperidin-3-amine
N-(propan-2-yl)-1-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
4-ethyl-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,2,3-thiadiazole-5-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
N,5-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2-methoxy-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-(3-hydroxypiperidin-1-yl)ethan-1-one
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide