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(2S,4R)-N-methyl-4-[(naphthalen-1-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-{[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzoic acid
3-{5-[2-(4-fluorophenoxy)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-methanesulfonamidopropanamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(3-methylpyridin-4-yl)piperazine
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
(2S,4S)-4-{4-[(1-adamantan-1-yl-N-methylformamido)methyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
2-amino-4-[5-(oxan-2-yl)furan-2-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
(3aR,6aR)-2-cyclopentyl-5-(2-methanesulfonamidoacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}but-2-ynamide
2-[3-(methoxymethyl)piperidin-1-yl]-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
2-methyl-3-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
5,7-dimethyl-N,N-dipropyl-2-(pyrimidin-5-yl)quinoline-4-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methylfuran-2-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
(1S,5R)-6-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-4-[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-yl]pyrimidine
4-[(3-acetamidopyrrolidin-1-yl)methyl]-N-(1-ethyl-1H-1,2,4-triazol-5-yl)benzamide
3-cyclohexyl-N-(2,2,2-trifluoroethyl)-1H-pyrazole-4-carboxamide
1-(5-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1H-1,2,4-triazol-1-yl)butan-2-ol
3-chloro-N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}benzamide
(1S,5R)-3-(2-methoxy-4-methylbenzenesulfonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-4H-chromen-4-one
2-amino-1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-methylpropan-1-one
N-methyl-2-(1-propylpiperidin-4-yl)-N-[1-(pyridin-3-yl)propyl]acetamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[2-(dimethylamino)ethyl]-3-ethylurea
1-methyl-4-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
2-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
3,3-dimethyl-1-(2-oxo-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)urea
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)-1-methylpiperidine-2-carboxamide
1-acetyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(1H-imidazol-1-yl)propan-1-one
5-ethanesulfonamido-1-methyl-2-phenyl-N-[2-(pyrazin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-methyl-N-[2-(oxan-2-yl)ethyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
1-[2-methoxy-4-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
3-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]propane-2-sulfonamide
N-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(methylsulfanyl)acetamide
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(thiophene-2-carbonyl)pyrrolidine-2-carboxamide
2-(3-methoxypropyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine
1-ethyl-5-(1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)-1H-1,2,4-triazole
2-ethyl-8-(5-propyl-1,2-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-{[(2-ethoxyphenyl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
[4-methyl-5-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methanol
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-N-cycloheptylpiperidine-1-carboxamide
2-{1-[4-(1H-pyrazol-3-yl)benzoyl]azetidin-3-yl}pyridine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2-methylfuran-3-carbonyl)piperidine-3-carboxylate
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]quinoline-2-carboxamide