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4-{methyl[(2E)-3-phenylprop-2-en-1-yl]amino}pyrimidine-5-carboxylic acid
5-(2-{2-[(4-aminopyrimidin-2-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
(3S,4R)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(thiophen-3-yl)phenoxy}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
1-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propane-1,2-dione
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-5-methoxy-3-methyl-1H-indole
2-[3-(1H-imidazol-1-yl)propyl]-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(3-methoxyphenyl)-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-{1-[4-(furan-2-yl)butan-2-yl]-1H-imidazol-2-yl}-2-methoxyphenol
2-(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}furan-2-yl)benzonitrile
4-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(1'-{[4-(2-aminoethyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)-2-methoxyethan-1-one
({1-[(1-hexylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)urea
methyl 1-ethoxy-8-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
5-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2-methoxyphenol
3-{1-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperidin-4-yl}benzonitrile
1-(piperidin-3-ylmethyl)-N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-3-(thiophen-2-yl)propan-1-one
3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}benzoic acid
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N,1-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-({1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}methyl)morpholine
2-[(1S,5R)-3-[(2-fluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
ethyl 1-(cyclopent-1-ene-1-carbonyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
1-[(4-methylphenyl)methyl]-3-(oxolan-3-yl)-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazole
methyl 3-(2H-1,3-benzodioxol-4-ylmethyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-fluorophenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}cyclopropane-1-carboxamide
[(2-fluoro-4-methoxyphenyl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
2-{4-[(2-methyl-1,3-thiazol-5-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
3-({1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}amino)pyrrolidin-2-one
(3aR,6aR)-2-cyclopentyl-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-cyclooctyl-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
5-(4-methoxyphenyl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1,2,4-triazin-3-amine
methyl 1-({4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
7-[(3-methoxyphenyl)methyl]-2-(4-methylpentanoyl)-2,7-diazaspiro[4.5]decan-6-one
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-2-methylpyrimidine-5-carboxamide
methyl 2-({[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-4-{1H-imidazo[4,5-b]pyridin-2-yl}-1H-pyrazole
2-amino-4-[4-(piperidin-1-ylmethyl)thiophen-2-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
5-chloro-2-methyl-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]benzamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
3-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetamido}-4-chloro-N,N-diethylbenzamide
N-{[7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2,5-dimethylfuran-3-carboxamide
6-(2-chlorophenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one