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N-(pyridin-3-ylmethyl)-1-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-benzyl-5-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione
9-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}-3-azaspiro[5.5]undecane
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
2-[2-(1H-pyrazol-1-yl)ethyl]-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
1-[3-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]ethan-1-one
3-[(2R,3R,6R)-5-(5-methoxyfuran-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
7-(2,2-dimethyloxane-4-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-{[1-butyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
N-[2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-4-methoxybenzene-1-sulfonamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyrrolidine-1-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-1-one
3-{[(3,4-dimethoxyphenyl)methyl]amino}-N-(thiophen-2-ylmethyl)propanamide
2,6-dihydroxy-N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]benzamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-methyl-2-phenylpropan-1-one
2-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carboxylic acid
N-cycloheptyl-3-{[(4-sulfamoylphenyl)methyl]amino}propanamide
(1R,3s,6r,8S)-4-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
(3S,4R)-4-methyl-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidine-3,4-diol
1-ethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{4-[(4-ethynylphenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-[3-(1H-1,2,3-triazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[(dimethyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-yl}methyl)butanamide
2-{4-[(butylcarbamoyl)amino]phenyl}-2-(thiomorpholin-4-yl)acetic acid
4-chloro-1-methyl-3-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}-1H-indazole
4-(naphthalen-2-yloxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
1-(adamantan-1-yl)-4-(1H-pyrrole-3-carbonyl)piperazine
2-[(2-methylphenyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(thiophen-2-yl)propanoyl]piperidine-2-carboxamide
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylacetamide
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
2-{4-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-6-(2-methyl-1,3-thiazol-4-yl)-3,4-dihydropyrimidin-4-one
4-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,4-oxazepane
1-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-2-(pyridin-3-yloxy)ethan-1-one
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)(2-phenoxyethyl)amine
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[2-(1,3-thiazol-4-yl)ethyl]urea
(1R,5S,6R,7S)-N,3-dimethyl-4-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-chloro-4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenol
2-[3-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)phenyl]ethan-1-amine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-methyl-5-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-1,2,4-oxadiazole
(3S,4S)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
1-(2-methoxyacetyl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}piperidine-4-carboxamide
N,N-dimethyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
(3R,4R)-4-ethyl-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine-3,4-diol
1-(2-ethoxyethyl)-5-(thiomorpholine-4-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one