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N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-methyl-1H-indole-3-carboxamide
N-methyl-2-[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]pyridine-4-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[1-(thiophene-3-carbonyl)piperidin-3-yl]propanamide
1-[(3-methylphenyl)methyl]-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazine
N-(cyclopropylmethyl)-4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-cyclopentyl-N-[3-(4-{[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}piperidin-1-yl)phenyl]acetamide
2-amino-6-cyclopropyl-4-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]pyridine-3-carbonitrile
1-{5-[(6-aminopyrimidin-4-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
1-(3-fluorophenyl)-3-(1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
7-(2-methoxyethyl)-2-[2-(thiophen-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2,5,6,7,8-hexahydroquinolin-2-one
4-{2-azaspiro[4.4]nonan-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
2-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
(3S)-1-[5-(2,3-dihydro-1H-isoindole-2-carbonyl)-1-methyl-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
8-[2-(4-chlorophenyl)morpholin-4-yl]-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
1-(propan-2-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
(2S,4S)-4-(2-chlorobenzamido)-1-methyl-N-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
3-[1-(difluoromethyl)-5-methyl-1H-pyrazol-4-yl]-N,N-dimethylaniline
3-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
N-{3-[(diethylamino)methyl]phenyl}-3-oxo-4-phenylpiperazine-1-carboxamide
N-(2-methoxyethyl)-3,5-dimethyl-4-oxo-N-(oxolan-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1-[(2-fluorophenyl)methyl]piperazin-2-one
(3aS,6aS)-5-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}-1-methyl-octahydropyrrolo[3,4-b]pyrrole
4-ethyl-N,N-dimethyl-6-(4-{[(5-methylpyrazin-2-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-amine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}-6-fluoro-1H-1,3-benzodiazole
(1R,4R)-2-{[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
2-[({3-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)(methyl)amino]-N-methylacetamide
1-cyclopentyl-N3-[3-(dimethylamino)-2,2-dimethylpropyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(1R,5R)-3-[2-(1H-imidazol-2-yl)benzoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
2-[(1-benzyl-1H-imidazol-2-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-{2-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]quinolin-6-yl}acetamide
5-(3,6-dimethylpyrazin-2-yl)-1,2,3,4-tetrahydroisoquinoline
N-cyclohexyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-1H-1,2,3-triazole-5-carboxamide
1-(6-cyanopyridin-3-yl)-3-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]urea
1-{3-[(diethylamino)methyl]phenyl}-3-(1H-pyrazol-3-ylmethyl)urea
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
N-(3-chloro-4-methoxyphenyl)-3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}propanamide
4-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
4-(4-fluorophenyl)-1-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperidin-4-ol
6-(2-methoxypyridine-3-carbonyl)-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-{[4-(methylsulfanyl)phenyl]methyl}-4-(piperidin-3-yl)-N-propylbenzamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-4-yl)propan-1-one
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-(2-chlorophenyl)propanamide
N-(1H-imidazol-2-ylmethyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-(1-ethyl-5-oxopyrrolidin-3-yl)-1,3-oxazole-4-carboxamide