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N-{1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperidin-4-yl}methanesulfonamide
2-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}-4-(6-methoxypyridin-2-yl)phenol
1-(2,2-dimethylpropyl)-4-{[(2-fluoro-5-methoxyphenyl)methyl]amino}pyrrolidin-2-one
1-[(2-methoxyphenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
{[(3S,4R)-1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-methyl-6-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)pyrimidin-4-ol
9-{[5-(hydroxymethyl)furan-2-yl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]acetamide
4-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
(2,3-dihydro-1-benzofuran-5-ylmethyl)({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(2-methoxyphenyl)ethan-1-one
3-chloro-5-[4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
4-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
4-(2-aminopyrimidin-4-yl)-7-(5-chloropyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-{1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)-1,3-thiazole
methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl](1,3-thiazol-4-ylmethyl)amine
1-{[5-(4-methanesulfonylphenoxy)-2-methoxyphenyl]methyl}pyrrolidine
5-ethyl-N4-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}pyrimidine-2,4-diamine
N-{[8-(propan-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-chloro-6-methoxy-3-(1-methyl-1H-1,3-benzodiazol-2-yl)phenol
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-4-oxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3-carboxamide
1-(3-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
3-{[(5-methylpyrazin-2-yl)methyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
2-(1H-1,3-benzodiazol-1-yl)-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-(2-methoxyphenoxy)acetamide
N-(2-hydroxyethyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[(3-methoxyphenyl)amino]butanamide
4-(8-hydroxyquinolin-2-yl)-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2,2-dimethyl-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-(3-hydroxypropyl)-2-methyl-N-[(5-methylthiophen-2-yl)methyl]-1,8-naphthyridine-3-carboxamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
7-(2,6-dimethoxyphenyl)-1,2,3,4-tetrahydroisoquinoline
1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
6-fluoro-2-({[(1-hydroxycyclohexyl)methyl]amino}methyl)quinolin-4-ol
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(pyrrolidin-1-yl)pyridazine
6-[({2-amino-6-[(4-methylphenyl)sulfanyl]pyrimidin-4-yl}amino)methyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-[2-(1H-indol-1-yl)ethyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-3,3-dimethylurea
(2R,6S)-1-(3-methyl-1H-pyrazole-5-carbonyl)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-ethyl-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-(cyclopropylmethyl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
6-methyl-N4-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidine-2,4-diamine
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
1-cyclopentyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
1-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one